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2-amino-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-6-(propan-2-yl)pyrimidine-4-carboxamide
4-[(4-fluorophenyl)methyl]-1-(5-methoxyfuran-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2,5-dioxo-6-[3-(2-propoxyphenyl)propyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-butoxy-1-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]ethan-1-one
(4S)-1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3,3,4-trimethylpiperidin-4-ol
1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-[3-({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propyl]piperidin-3-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
[(3R,4R)-1-{[5-(4-methylphenyl)furan-2-yl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2-chloropyridin-3-yl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
4-[(4-fluorophenyl)methyl]-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,1,3-trimethyl-N-(1-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-5-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]pyrrolidine-3-carboxylic acid
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[3-(methylsulfanyl)phenyl]urea
4-methyl-2-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-5,6,7,8-tetrahydroquinazoline
4-ethyl-3-(2-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-4H-1,2,4-triazole
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
(4aS,8aS)-2-[4-(trifluoromethyl)pyridin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
N-cyclopentyl-N-({4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-4-(1H-pyrazol-1-yl)benzamide
3-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]azetidin-3-yl}pyridine
2-amino-7-[6-(propan-2-yl)-1H-indole-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(2-methoxyphenyl)ethyl]-6-[(4-phenylphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-[1-methyl-4-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)piperazin-2-yl]ethan-1-ol
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylate
10-methoxy-5-[3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-(1-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
5-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
(3R,4R)-1-(3-chlorothiophene-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-(propan-2-yl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidine
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pentan-1-one
N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}oxolane-2-carboxamide
N,2-dimethyl-6-(piperidin-3-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
(3aS,6aS)-2-benzyl-5-(1,4-dithiepan-6-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-chlorophenyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]-5-methylpiperazin-2-one
N-[2-(4-methoxyphenyl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-cyclopropyl-N-[(2-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}azocane
{3-[(2-fluorophenyl)methyl]-1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]piperidin-3-yl}methanol
N-[(5-methylpyrazin-2-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
6-ethyl-5-methyl-N4-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidine-2,4-diamine
(3S,4S)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](furan-2-ylmethyl)(3-methylbutan-2-yl)amine
4-(hydroxymethyl)-1-(2-methyl-1-benzofuran-5-carbonyl)azepan-4-ol
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(morpholin-4-yl)piperidin-1-yl]ethan-1-one