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1-(2-methoxyethyl)-N3-[(4-methylphenyl)methyl]-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-{2-[2-(3-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-2,6-dimethyl-1,4-dihydropyridin-4-one
7-(2-hydroxyethyl)-2-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2,3-dihydro-1H-inden-2-yl)-3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-{4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]phenyl}acetamide
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
5-[butyl(methyl)amino]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N'-(2,4-dimethylphenyl)-N-[2-(dimethylsulfamoyl)ethyl]ethanediamide
[3-(1H-1,2,3-benzotriazol-1-yl)propyl]({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[2-(methylsulfanyl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-methyl-2-(1-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
3-cyclopropyl-1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]propan-1-one
1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-[3-(dimethylamino)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-(2,3-dihydro-1H-isoindol-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
N-methyl-N-(propan-2-yl)-2-[2-(pyridin-2-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(3aS,6aR)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[1-(5-fluoropyridine-3-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
N-[(3R,4R)-3-hydroxy-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl]pyridine-2-carboxamide
N3-benzyl-1-cyclopentyl-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]oxane-4-carboxamide
3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-6-(quinolin-5-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-chloro-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxypropanamide
4-(benzyloxy)-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
N-(3-ethylphenyl)-4-oxo-4-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}butanamide
2-cyclopropyl-9-(4-oxo-4-phenylbutyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-N3,N3-diethyl-N5-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{1-[4-(hydroxymethyl)benzoyl]piperidin-3-yl}-3-phenylpropan-1-one
N-[2-(ethanesulfonyl)ethyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)benzonitrile
3-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-chloro-1-ethyl-1H-pyrazole
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)propyl]piperidin-4-ol
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
(2S,4R)-4-(benzylamino)-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
3-{1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-cyclobutyl-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
[(8-methoxyquinolin-5-yl)methyl](methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-[3-(1,3-oxazol-5-yl)phenyl]piperazine-1-carboxamide
N-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
3-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
1-{5-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
1,2-dimethyl-3-[4-(pyridin-4-yl)piperazine-1-carbonyl]-1H-indol-5-ol
N-cyclopropyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-{[2-(1H-imidazol-4-yl)ethyl]sulfamoyl}-N-(3-methylbutan-2-yl)benzamide
1,4-dimethyl-9-[3-(5-methylfuran-2-yl)butyl]-1,4,9-triazaspiro[5.5]undecane
2-(5-acetylthiophen-3-yl)-N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]acetamide