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(2,4,6-trimethyl-3-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenyl)methyl acetate
1-[2-methoxy-5-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-[4-(1,4-dithiepan-6-yl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
2,4-dimethyl-6-[3-(2-phenylethyl)piperidine-1-carbonyl]pyrimidine
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)acetamide
N-cyclopentyl-1-[1-(3-methylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(1H-pyrrole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
methyl 1-ethoxy-8-[2-(methoxycarbonyl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-5-phenyl-1,2-oxazole-3-carboxamide
4-[(4aS,7aR)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
2-[3,5-dimethyl-4-(2,2,2-trifluoroethanesulfonamido)-1H-pyrazol-1-yl]acetic acid
1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
8-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
dimethyl[(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)sulfamoyl]amine
1-(3-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)pyrrolidin-2-one
(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanamine
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
3,5-dichloro-N-ethyl-4-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
3-[2-({1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrrol-1-yl]pyridine
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
5-{[3-(4-benzylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-2-methylpyridine
N,N,4-trimethyl-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]pyrimidin-2-amine
2-methyl-6-[2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]pyrimidin-4-ol
N-[(5-methoxy-1H-indol-2-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
3-ethyl-8-[(2-hydroxynaphthalen-1-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1,3-dihydroxypropan-2-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
3-(cyclobutylmethyl)-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-(oxolan-2-ylmethyl)urea
N,N-diethyl-2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}acetamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
7-(1,3-benzothiazol-2-yl)-4-[(3,4-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 1-[6-(dimethylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidine-4-carboxylate
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]oxolane-2-carboxamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-{[3-(morpholin-4-yl)phenyl]methyl}piperidin-4-ol
{6-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}methanol
2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(pyridin-2-yl)ethyl]acetamide
7-(2-cyclohexylethyl)-2-(propane-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(2-methoxyphenyl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]furan-2-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidine-2-carboxamide
(2S,4S)-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-1-(2-methylpropyl)pyrrolidine-2-carboxamide
N-[(2-methoxyphenyl)methyl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
(4aS,7aR)-1-(2-ethoxyacetyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-ethyl-N-[1-(pyrazin-2-yl)propan-2-yl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(propan-2-yl)acetamide
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-(pyrrolidin-1-yl)butan-1-one
5-{1-[2-(3-chlorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
5-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-2-(3-methylphenyl)pyrimidine
N-[(4-fluorophenyl)methyl]-3-[1-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)piperidin-4-yl]propanamide