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4-{[1-(carbamoylmethyl)piperidin-4-yl]oxy}-3-chloro-N-[2-(dimethylamino)ethyl]benzamide
3-{[2-(4-fluorophenyl)pyrrolidin-1-yl]sulfonyl}pyridine
2-{1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl}-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
1-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-4-carboxamide
1-(2-fluorophenyl)-N-(3-hydroxypropyl)-2,2-dimethyl-N-(pyridin-4-ylmethyl)cyclopropane-1-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-(2-propoxyacetyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}acetamide
{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
5-methyl-3-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-{[1-(1H-indol-2-yl)ethyl](methyl)amino}-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]acetamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(3-sulfamoylphenyl)piperidine-1-carboxamide
N-ethyl-3,4,7-trimethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-indole-2-carboxamide
ethyl 1-(cyclopropylmethyl)-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2,2-dimethyloxan-4-yl)-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
{5-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
methyl 2-[2-(1-benzyl-3-oxopiperazin-2-yl)-N-methylacetamido]acetate
N,N-dimethyl-4-oxo-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butanamide
N-{[4-(3-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
1-(3-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(quinolin-2-ylmethyl)amine
(1R,5S,6S)-6-{[4-(3-fluorophenoxy)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)urea
ethyl 2-[1-(1-cycloheptyl-6-oxopiperidin-3-yl)-N-methylformamido]acetate
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]phenol
(2S)-2-(methoxymethyl)-N-(1,2,3-thiadiazol-5-yl)pyrrolidine-1-carboxamide
(1S,4S)-2-(3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)-2-azabicyclo[2.2.1]heptane
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-{imidazo[1,2-a]pyridin-2-yl}-N-methylpropanamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-4-(quinoxalin-5-ylmethyl)-1,4-diazepan-2-one
1-{3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
2,2-dimethyl-1-{6-methyl-5-[5-(pyridin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}propan-1-one
(3aR,7aS)-2-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-[(5-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-methylpiperidine
2-{5-[(1S)-1-hydroxy-2-phenylethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
N-methyl-2-(5-oxo-2-phenylcyclopent-1-en-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
(3S,4R)-1-(3-chloropyridin-2-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
N-(1-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
4-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
4-[(1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}piperidin-3-yl)methyl]morpholine
(3S,4S)-N-(3,5-dichlorophenyl)-3-hydroxy-4-(piperidin-1-yl)pyrrolidine-1-carboxamide
methyl 2-{1-[2-(cycloheptylcarbamoyl)ethyl]-3-oxopiperazin-2-yl}acetate
1-{2-hydroxy-3-[4-methoxy-2-(pyrrolidin-1-ylmethyl)phenoxy]propyl}piperidin-4-ol
2-{2-[2-(1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
N-ethyl-2-hydroxy-4-(methylsulfanyl)-N-[2-(1H-pyrazol-1-yl)ethyl]butanamide
3-(4-fluorophenyl)-N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide