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1-{5-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]thiophen-2-yl}ethan-1-one
6-[2-(furan-2-yl)azepane-1-carbonyl]-2,3-dimethylquinoxaline
N-[2-(4-sulfamoylphenyl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-(pyridin-3-ylmethyl)-4-{[3-({1-[2-(trifluoromethoxy)benzenesulfonyl]piperidin-4-yl}oxy)phenyl]methyl}piperazine
4-[(2-cyclohexylpyrimidin-5-yl)methyl]piperazine-1-sulfonamide
1-[3-(furan-2-yl)phenyl]-N-(1-propylpiperidin-4-yl)piperidin-4-amine
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-ethyl-1-methyl-3-{[1-(2-methyl-1H-imidazole-4-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{2-[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]ethyl}benzoic acid
4-(adamantane-1-carbonyl)-2-benzylmorpholine
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
N'-[(4-chlorophenyl)methyl]-N'-ethyl-N-(1,3,4-thiadiazol-2-yl)ethanediamide
3-[(2-fluorophenyl)methyl]-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2-(trifluoromethyl)benzamide
2-(2-hydroxyethyl)-8-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[2-(1H-pyrazol-4-yl)ethyl]-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]ethan-1-one
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(3-methoxyphenyl)-1-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl]-N,3-dimethylbutanamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}quinoline
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4,4,4-trifluorobutanamide
methyl 2-{4-[4-(piperidin-3-yl)benzamido]piperidin-1-yl}acetate
3-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-1-(oxan-4-yl)urea
5-(3-methoxyphenyl)-4-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)pyrimidine
1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
1-[(4-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)-N-(3-methoxyphenyl)piperidine-1-carboxamide
1-(2-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}ethyl)imidazolidin-2-one
N-ethyl-2-{3-[3-(pyridin-4-yl)phenyl]-1H-pyrazol-1-yl}acetamide
4-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}pyridine
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-methanesulfonyl-1,4-diazepane
3-{5-[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]-1,2,4-oxadiazol-3-yl}pyridazine
1-(furan-2-ylmethyl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxyacetamide
(1S,2R)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyrrolidine-1-carbonyl)cyclohexane-1-carboxamide
N-(5-chloro-2-ethyl-3-methyl-1-benzofuran-7-yl)-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
N-(1-{4-[4-(3,5-dimethylphenyl)-3-oxopiperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
(1R,5S,8R)-N,N-dimethyl-3-[(3-methylquinoxalin-2-yl)methyl]-3-azabicyclo[3.2.1]octan-8-amine
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(9H-purin-6-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S)-2-{[(cyclooctylcarbamoyl)methyl]amino}-3-methylbutanamide
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})amine
8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N,1-dimethylazepane-2-carboxamide
4-(benzyloxy)-1-(1,2-oxazole-3-carbonyl)piperidine
methyl 7-oxo-9-(3-phenylpropoxy)-3-[2-(thiophen-2-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate