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methyl 3-(2-fluorobenzoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
3-cyclohexyl-4-{[4-(1H-imidazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
4-benzyl-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-one
3-[1-(methoxymethyl)cyclopentyl]-1-[2-(trifluoromethyl)phenyl]urea
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl})methylamine
1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[1-(thiophen-2-yl)ethyl]piperidine-4-carboxamide
N4-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]pyrimidine-4,6-diamine
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(pyrazin-2-yl)ethyl]amine
7-chloro-4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2,5-dimethylphenyl)piperazine
8-[(2-tert-butyl-5-carbamoylfuran-3-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[(4-chlorophenyl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[4-(3-cyano-5,6,7,8-tetrahydroquinolin-2-yl)piperazin-1-yl]-N-ethylacetamide
(1R,2R,4R)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
4-benzyl-N-(3-chlorophenyl)-4-(hydroxymethyl)piperidine-1-carboxamide
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-hydroxypropan-1-one
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
N-(4-chloro-3-methylphenyl)-4-[3-(dimethylamino)-2-hydroxypropyl]piperazine-1-carboxamide
3-tert-butyl-1-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}urea
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)cyclopropan-1-amine
3-[3-(oxolan-3-yl)propyl]-1-[2-(trifluoromethyl)phenyl]urea
2-methyl-4-[4-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)phenyl]butan-2-ol
ethyl 1-[2-(4-hydroxypiperidin-1-yl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2H-1,3-benzodioxole-5-carboxamide
2-[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(morpholin-4-yl)ethan-1-one
2-({[(3R,4R)-1-(6-chloro-1,3-benzothiazol-2-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
(4aS,7aR)-1-(cyclopropanesulfonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-(4-fluorophenyl)-N-[3-(1H-imidazol-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[1-(4-fluorophenyl)propyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-(3-phenylpiperidin-1-yl)-N-[2-(pyridin-4-yl)ethyl]acetamide
5-(2-ethoxy-5-methylbenzenesulfonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl)amino)-2-(2,4,6-trimethylphenyl)acetic acid
2-{1-[(2-ethoxyphenyl)methyl]-4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-(diethylamino)-3-[5-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
5-(2,4-dimethoxyphenyl)-3-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-1,2,4-triazine
N-cyclopropyl-3-[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-4-yl]propanamide
1-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
ethyl 1-(3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperidine-4-carboxylate
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(1-methylpiperidin-2-yl)methyl]acetamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(4,4,4-trifluorobutyl)piperidine
1-ethyl-5-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,2,4-triazole
5-({1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-2,1,3-benzothiadiazole
2-(4-chlorophenyl)-4-(2,6-difluorobenzoyl)morpholine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxopiperidin-1-yl)acetamide
7-chloro-3-({methyl[1-(3-methylpyridin-2-yl)propan-2-yl]amino}methyl)-1,2-dihydroquinolin-2-one