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5-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-[6-(morpholine-4-carbonyl)pyrazin-2-yl]benzoic acid
methyl 3-(cyclobutylmethoxy)-5-[(2-hydroxy-2-methylpropyl)carbamoyl]benzoate
4,6-dimethyl-2-(pyridin-4-yl)pyridine-3-carboxamide
2-methyl-6-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamido}acetic acid
N-ethyl-3-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propanamide
3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(3R)-1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
4-chloro-1-ethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(2-ethoxypyridin-3-yl)-2-(4-methoxypiperidin-1-yl)acetic acid
(1S,5R)-6-(3,4-dimethylbenzoyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(3-methoxyphenyl)-N-{[4-(morpholin-4-yl)phenyl]methyl}acetamide
N-{[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
2-{4-[2-(morpholin-4-yl)-2-oxoethyl]-2-oxopiperazin-1-yl}benzonitrile
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
2-(2-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
N-(2H-1,3-benzodioxol-5-yl)-4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carboxamide
3-[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]propane-1,2-diol
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
(1S,5R)-6-[(3-chloro-4-methoxyphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-{2-[4-(1H-pyrazol-5-yl)phenyl]phenoxy}propanamide
N-{[3-methoxy-4-(pyridin-2-ylmethoxy)phenyl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-ethyl-2-(2-ethylpyrimidin-5-yl)-5,7-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
(2S)-N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-methyl-3-phenyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(pyridin-2-yl)acetamide
2-[2-(dimethylamino)ethyl]-9-[2-hydroxy-2-(4-methoxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-2-{[1-(1-ethylpiperidin-4-yl)piperidin-4-yl]oxy}-4-methoxybenzamide
4-benzyl-3-ethyl-1-(3-fluoro-4-methylbenzoyl)-1,4-diazepan-5-one
1-[2-(dimethylamino)ethyl]-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(2-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}benzamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-fluoro-4-methylbenzamide
4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
5-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
4-[2-(dimethylamino)ethoxy]-N-[2-methoxy-5-(methylcarbamoyl)phenyl]piperidine-1-carboxamide
1-(2-hydroxyethyl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]piperidine-4-carboxamide
(3S,4R)-N,N-dimethyl-4-propyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-amine
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
1-(2-{[4-(2-hydroxyethyl)piperidin-1-yl]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
9-methoxy-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-ethyl-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
N-cyclopropyl-6-(2,5-dimethylfuran-3-yl)-7-methyl-N-(2-methylpropyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}pyridine-3-carboxamide