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1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-4-(thian-4-yl)piperazine
7-[(2,3-difluorophenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decane
(1S,5R)-3-benzoyl-N-(2,4-dimethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-{1-[1-(propane-1-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
5-{2-[2-(2-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}-1H-1,2,3-benzotriazole
4-(cycloheptylsulfamoyl)-N-(oxolan-3-yl)benzamide
1-cycloheptyl-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-(4-tert-butylbenzoyl)-4-methyl-1,4-diazepan-5-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,3-dimethoxybenzamide
1-{3,5-dimethyl-4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
6-(2-chlorophenyl)-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N,2-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[(3S,4R)-1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(3,4,5-trifluorophenyl)methyl]pyrrolidin-3-yl]methanol
1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclohexan-1-ol
(1S,5R)-3-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-benzyl-5-[1-(2-methylbutanoyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
(1S,5R)-6-(2-methoxyethyl)-3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonane
N-(1-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
(3S,4S)-4-cyclopropyl-1-(2,5-dimethylfuran-3-carbonyl)pyrrolidine-3-carboxylic acid
(2S,4S)-4-amino-1-(4-chloro-3-methylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 5-[(1-methyl-1H-indol-3-yl)methyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(6-cyanopyridin-3-yl)-4-{[2-(2-hydroxyethyl)piperidin-1-yl]methyl}benzamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-(4-methylpiperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{4-[(4-methoxy-2,3-dimethylphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(6-methoxypyrimidin-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-methyl-7-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-[4-({ethyl[(1R,2R)-2-hydroxycyclohexyl]amino}methyl)phenyl]-6-propyl-3,4-dihydropyrimidin-4-one
N-{[1-(3-phenoxypropyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}acetamide
methyl 5-[2-(6-chloropyridin-3-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
6-{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-9H-purine
2-[methyl({4-methyl-5-[1-(pyridine-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
methyl[(1-phenylpyrrolidin-3-yl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
2-[2-(3-methoxyphenoxy)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(2-methoxyphenyl)methyl]piperazine
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(isoquinoline-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-benzyl-1-(2-phenylethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[4-(2-methoxyphenyl)-5-(1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-(3-hydroxy-3-methylbutyl)-N-[1-(hydroxymethyl)cyclohexyl]benzamide
6-[(3-methoxyphenyl)methoxy]-4-(5-methyl-1H-pyrazole-3-carbonyl)-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
(3R,4S)-4-(5-methylfuran-2-yl)-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-amine
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-(1-{7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
1-[3-(difluoromethoxy)benzoyl]-4-(pyrrolidine-1-carbonyl)piperidine
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-6-(3-methoxyphenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3-methylpiperidine