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ethyl 2-{[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]amino}acetate
N-(2-methoxyethyl)-N-methyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
8-[(cyclohexylmethyl)carbamoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperazine
9-methoxy-7-(pyridin-3-yl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-(2,6-dimethylpyridin-4-yl)piperazine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine
1-ethyl-3-(2-methylpropyl)-N-[(1s,4s)-4-aminocyclohexyl]-1H-pyrazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-5-[(5-methylthiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)methyl]acetamide
1-(2-cyclohexylethyl)-N-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
methyl (2S,4R)-1-[(2-ethoxyphenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
1-(4-methanesulfonylphenyl)-3-phenyl-5-(1H-pyrazol-3-yl)-1H-1,2,4-triazole
(3aR,5R,6S,7aS)-2-(2,6-difluoro-3-methoxybenzoyl)-octahydro-1H-isoindole-5,6-diol
4-{2-[(3-methoxyphenyl)methyl]morpholine-4-carbonyl}benzene-1-sulfonamide
3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-5-(pyrrolidine-1-carbonyl)-1,2-oxazole
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-(1-methyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-({7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
1-(2-{2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-4-yl}-2-oxoethyl)-1,2,3,4-tetrahydroquinolin-2-one
N-[(1S,2R)-2-[(1-acetylpiperidin-4-yl)amino]cyclobutyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-2-(methoxymethyl)piperidine
3-{1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-(1-methyl-1H-pyrazol-3-yl)piperidine
1-benzyl-6-(pyridin-3-ylmethoxy)-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-2-one
5-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-1H-indole
4-{1-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]azetidin-3-yl}pyridine
N-(1,3-benzothiazol-2-ylmethyl)-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
3-methyl-4-(1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
3-(2H-1,3-benzodioxol-5-yl)-5-[(4-methoxyphenyl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-{1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
(3R,4S)-4-(3-methoxyphenyl)-1-(9H-purin-6-yl)pyrrolidin-3-amine
2-[3-(1H-indol-3-yl)-5-(morpholin-3-ylmethyl)-1H-1,2,4-triazol-1-yl]acetic acid
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(1,2-oxazinan-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
4-(2-acetylphenyl)-N-(prop-2-en-1-yl)benzamide
9-[2-(3-ethyl-2-imino-2,3-dihydro-1H-1,3-benzodiazol-1-yl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
(3R,5S)-N3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
methyl 4-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-oxobutanoate
3-{[1-(2,5-dimethylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
1-methyl-1'-(3-phenyl-1H-pyrazole-4-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-{1-[1-(2,2-diphenylethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-(1-ethylpiperidin-4-yl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N-[2-({2-cyclopentyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-N-methylmethanesulfonamide
5-[1-(2,2-dimethylpropyl)-4-hydroxypiperidin-4-yl]-N-methyl-N-(quinolin-5-ylmethyl)-1-benzofuran-2-carboxamide
1,3-dimethyl-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-(5-ethyl-2-methylpyrimidin-4-yl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-cycloheptyl-4-oxo-1-(propan-2-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide