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N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
N-(3-chloro-4-fluorophenyl)-3-{1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}propanamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
5-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}isoquinoline
2-(3-methanesulfonylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[1-(3,4-dimethylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]pyridazine
3-cyclopropyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-pyrazole-5-carboxamide
(3S,4R)-3-acetamido-4-(4-methoxyphenyl)-N-[(2-methylphenyl)methyl]pyrrolidine-1-carboxamide
5,7-dimethyl-N-[3-(morpholin-4-yl)propyl]pyrido[2,3-d]pyrimidin-4-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-3-phenylpyrrolidine-2,5-dione
2-{3-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
2-(2-phenylethyl)-N-[1-(pyrimidin-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-2-[4-(quinolin-2-yl)-1H-pyrazol-1-yl]acetamide
1-(4-fluorophenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3,5-dimethyl-1H-pyrazole
(2S,4R)-1-[(4-chlorophenyl)methyl]-N,N-diethyl-4-{[(2-hydroxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-(2-methoxy-5-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
5-(4-acetylpiperazine-1-carbonyl)-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanamide
(3S,4S)-1-phenylmethanesulfonyl-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-(4-methoxyphenyl)-N-({1-[2-(pyrrolidin-1-yl)acetyl]piperidin-3-yl}methyl)acetamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(2-fluorophenyl)methyl]piperidine
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)quinoline-8-sulfonamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
2-[3-(methylcarbamoyl)phenyl]-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
4-(1-benzothiophen-3-yl)-6-methyl-2,3-dihydropyridazin-3-one
3-[2-(furan-2-yl)azepane-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
3-[2-(4-fluorophenyl)ethyl]piperidine
3-[2-(2,5-dichlorophenyl)-1H-imidazol-1-yl]benzamide
3-{1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidin-3-yl}benzoic acid
8-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(2S,4R)-4-{[(2,6-difluorophenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
1-{4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]thiophen-2-yl}ethan-1-one
2-{4-methyl-6-[3-(morpholin-4-yl)azetidin-1-yl]pyrimidin-2-yl}phenol
2-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-6-methylquinolin-4-ol
9-(quinolin-4-ylmethyl)-3,9-diazaspiro[5.6]dodecane
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 1-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxylate
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-(3-chloro-4-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)cyclopentanecarboxamide
methyl 3-acetamido-1-ethyl-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-methoxy-8-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(morpholine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1-{1-[3-(3-methylphenyl)phenyl]piperidin-4-yl}pyrrolidin-3-yl)acetamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-1,1-dioxo-1λ6-thiolane-3-carboxamide
2-methyl-4-[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane-6-carbonyl]quinoline
3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-phenylpiperidine-1-carboxamide
ethyl 5-(1-ethyl-1H-pyrazole-4-carbonyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(4-tert-butylphenoxymethyl)-5-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}pyrimidin-4-ol
N'1-ethyl-N'1-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopropane-1,1-dicarboxamide