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5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)pyridin-2-amine
4-(2-{3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}ethyl)benzene-1-sulfonamide
(3R,4S)-4-cyclopropyl-1-(5-methoxy-1H-indole-2-carbonyl)pyrrolidin-3-amine
2-(2-chlorophenoxy)-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}acetamide
N-benzyl-N-(oxolan-2-ylmethyl)-5-propyl-1,2-oxazole-3-carboxamide
(3R,4R)-3-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-3-hydroxy-4-methylpyrrolidine-1-carboxamide
9-(2,3-dihydro-1H-indene-1-carbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-phenylpyrrolidin-2-one
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-[1,2,3]triazolo[4,5-b]pyridine
5-(4-fluorophenyl)-2-methyl-4-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]pyrimidine
3-(3-methoxyphenoxy)-1-[4-(trifluoromethyl)benzoyl]azetidine
(1-{[(1H-indol-4-ylmethyl)(methyl)amino]methyl}cyclopentyl)methanol
1-(3-methoxyphenyl)-5-methyl-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamide
N-[2-(2-fluorophenoxy)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
6-phenyl-2-{2-[2-(thiophen-2-yl)-1H-imidazol-1-yl]ethyl}-2,3-dihydropyridazin-3-one
N-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-N-methyloxan-4-amine
(1R,9aR)-1-({[(2,5-dimethylphenyl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-1-methyl-3-({[(3-methylphenyl)methyl]amino}methyl)piperidin-2-one
N-(2-hydroxyethyl)-3-(4-hydroxyphenyl)-N-[(5-methylthiophen-2-yl)methyl]benzamide
1-(4,7-dimethylquinazolin-2-yl)-N-[(3-methoxyphenyl)methyl]piperidine-4-carboxamide
9-(2-methylbenzenesulfonyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-4-oxo-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,4-dihydropyridine-3-carboxamide
2-(cyclohexylmethyl)-4-(2,3-dimethoxybenzoyl)morpholine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
(1S,5R)-6-benzyl-3-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(ethoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
N2-benzyl-N2,7,7-trimethyl-N5-[4-(methylamino)pyrimidin-2-yl]-5,6,7,8-tetrahydroquinazoline-2,5-diamine
11-acetyl-4-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(1,3-thiazol-4-ylmethyl)piperidine
N-(2-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}ethyl)pyrimidine-5-carboxamide
3-(3-fluorophenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
2-ethyl-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1-[2-(1H-pyrazol-4-yl)ethyl]-1H-imidazole
1-[2-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-cyclopentyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-5-methylthiophene-2-carboxamide
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
(2S,4R)-1-[(4-ethylphenyl)methyl]-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
5-{[(3-fluorophenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-methyl-2-(4-phenylphenyl)-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
7-[(3,4-difluorophenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
5-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
1'-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(pyridin-2-yl)-7-[2-(pyrrolidin-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylfuran-3-carboxamide
1-[(butan-2-yl)carbamoyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
3-(4-fluorophenoxymethyl)-1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidine
4-(6-methoxypyridazin-3-yl)-1H-indole