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1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
methyl 4-({2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
1-{4-[4-methoxy-2-(2-methyl-1,4-oxazepane-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]cyclopentanecarboxamide
2-amino-4-(3-chloro-4-hydroxyphenyl)-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-cyclopropyl-1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-methylimidazo[1,2-a]pyridine-2-carboxamide
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxylate
{5-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-2-ethoxyphenyl}methanol
4-(3-methyl-1-benzothiophen-2-yl)-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
6-{2-[1-(2,3-dihydro-1H-inden-2-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydropyridazin-3-one
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-(methoxymethyl)thiophene-2-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[3-(2-hydroxyethoxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[3-(2,6-dimethylphenoxy)azetidin-1-yl]pyridine
1-ethyl-N-[(4-fluorophenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-phenylpiperidin-4-ol
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-indazole-3-carboxamide
2-amino-4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrimidine-5-carboxamide
3-[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
3-(1H-indol-5-yl)-N,N-dimethylpyrazin-2-amine
N-methyl-N-[2-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)ethyl]methanesulfonamide
N-[(4-fluorophenyl)methyl]-1-methyl-N-(pyridin-2-ylmethyl)piperidine-2-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(2-phenylethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
N-cyclohexyl-5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-[2-(dimethylamino)ethyl]-8-(2,6-dimethylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(1-methylpiperidin-2-yl)methyl]benzamide
[4-(4-methoxy-2,6-dimethylphenyl)pyridin-2-yl]methanol
N-[(3,4-dimethoxyphenyl)methyl]-3-(3-fluorophenyl)-N-(pyridin-4-ylmethyl)benzamide
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
2-methyl-8-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(4aS,7aR)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-8-methoxy-1,2,3,4-tetrahydroquinolin-2-one
3-(oxolan-3-yl)-5-{2-[5-(thiophen-2-yl)furan-2-yl]ethyl}-1,2,4-oxadiazole
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2,2-diphenylethan-1-one
1-[(3-chlorophenyl)methyl]-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
1-[(4-fluorophenyl)methyl]-4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-2-one
1-(4-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
1-[3-(adamantan-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidine
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
1-[2-(1-{3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanoyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N,1-diethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
3-[N-(2-phenylethyl)-1-(2,3,6-trimethylquinolin-4-yl)formamido]propanamide
3-[(4aR,8aR)-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridine-1-carbonyl]-2,3-dihydro-1H-inden-1-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(2-methylpyrimidin-4-yl)piperidin-3-yl]propan-1-ol