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2-[methyl(pyridin-2-ylmethyl)amino]-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
4-(1H-imidazol-2-yl)-1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidine
ethyl 5-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
(1S,5R)-3-methyl-6-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2,2-dimethyloxane-4-carboxamide
(1R,5R)-3-benzoyl-6-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(2S)-1-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(4-methoxyphenoxymethyl)piperidine
3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-4-[(4-methylphenyl)methyl]piperazin-2-one
N-[(2R,3R)-2-methoxy-1'-(2-methylpropanoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-(6-cyanopyridin-3-yl)-3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)benzamide
6-fluoro-4-hydroxy-N-(1-hydroxybutan-2-yl)-N-(pyridin-4-ylmethyl)quinoline-3-carboxamide
7,7-dimethyl-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-methyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazol-2-yl}-2,1,3-benzothiadiazole
N-[(2R,3R)-2-(benzyloxy)-1'-(quinoxalin-5-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
4-{[5-(diethylamino)pentan-2-yl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
3-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
2-methyl-4-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}pyrimidine
4-(1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}piperidin-3-yl)benzoic acid
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2,8-trimethylquinoline-4-carboxamide
methyl (2S)-1-[1-benzyl-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carbonyl]pyrrolidine-2-carboxylate
N-methyl-4-oxo-4-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
5-chloro-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-(9H-purin-6-yl)piperidin-4-amine
N-[(2-ethoxyphenyl)methyl]-N-ethyl-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-4-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]acetamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]amine
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetamide
dimethyl({[4-(2-methyl-5-propylpyrimidin-4-yl)-1,4-oxazepan-6-yl]methyl})amine
3-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
5-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]pyridine-3-carboxamide
ethyl 1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine-3-carboxylate
1-(2-ethoxyethyl)-2-oxo-N-(2,2,2-trifluoroethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-imidazole-2-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-[3-(morpholin-4-yl)propyl]piperidine-3,5-dicarboxamide
3-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
1,4-dimethyl-9-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1,4,9-triazaspiro[5.5]undecane
4'-(cyclobutylmethyl)-3'-oxo-N-(pyridin-3-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-carboxamide
{2-[4-(4-ethenylbenzoyl)morpholin-2-yl]ethyl}dimethylamine
8-[2-(4-methylphenoxy)acetyl]-2-phenyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-{2-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2,3-dihydro-1H-indazol-3-one
7-[(4-chlorophenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-methyl-1-(prop-2-en-1-yl)-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
2-cyclopentyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine