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5-benzyl-1-(3-chlorophenyl)-4-[2-(methylamino)acetyl]piperazin-2-one
3-cyclohexyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
3-[1-(3-chloropyridin-2-yl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
7-[2-(methylamino)pyridine-3-carbonyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
2-({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}amino)-6-methylpyridine-3-carbonitrile
(3R,4R)-3-hydroxy-N-(2-methylphenyl)-4-{[2-(3-methylpyridin-2-yl)ethyl]amino}pyrrolidine-1-carboxamide
4-(5-methylpyridin-2-yl)-1-(quinolin-2-yl)piperidin-4-ol
1-[2-(1,3-thiazol-2-yloxy)hex-5-en-1-yl]piperidine-4-carboxylic acid
1-(3-methoxy-4-{[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
2-(3-phenylpropyl)-8-(pyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-hydroxyethyl)-N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}piperidine-3-carboxamide
N-butyl-3-({[2-(1H-indol-1-yl)ethyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
[(3R,4R)-1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(2-methyl-1H-indol-1-yl)propanamide
5-[2-(difluoromethoxy)benzoyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
methyl 3-[2-(2-methoxyphenoxy)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1S,5R)-3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2,4-dimethyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidine
3-(4-methoxyphenyl)-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
4-chloro-2-[(3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]phenol
1-(2-{[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}-4-methylpyrimidin-5-yl)ethan-1-one
(2S)-1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-methyl-2-(propan-2-yl)piperazine
2-{4-[2-(dimethylamino)benzoyl]morpholin-3-yl}-N-(oxan-4-yl)acetamide
2-amino-6-(2-fluorophenyl)-4-(3-hydroxy-4-methoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(4-phenylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
[2H-1,3-benzodioxol-5-yl(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)methyl]dimethylamine
N-(2,3-dihydro-1H-inden-2-yl)-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-(2-hydroxyethyl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-1H-1,3-benzodiazole-5-carboxamide
2-(dimethylamino)-N-[2-(3-ethoxyphenoxy)ethyl]-N,4-dimethylpyrimidine-5-carboxamide
5-[(diethylcarbamoyl)methyl]-1-ethyl-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,N-bis(2-hydroxyethyl)-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
2-(2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}ethoxy)ethan-1-ol
1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-[(3-methylthiophen-2-yl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-sulfamoyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)benzamide
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
4-[(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methyl]morpholine
1-(4-ethylpiperazin-1-yl)-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propan-1-one
N,4-dimethyl-6-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-2-amine
(4aS,7aR)-1-[(2E)-hex-2-en-1-yl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]furan-2-yl}methanol
(3S,5R)-1-[(2,4-difluorophenyl)methyl]-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
(1R,5R)-N-(2-phenylethyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{4-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]piperazin-1-yl}-N-ethylacetamide
2-{[4-(6-ethoxy-4-methylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}phenol
3-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methoxy}pyridin-2-amine
N-[2-(3-methoxyphenyl)-1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)ethyl]-N-methylfuran-2-carboxamide