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1-[9-acetyl-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(3aS,6aR)-5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 9-[(1-methylpiperidin-3-yl)methoxy]-3-{[4-(methylsulfanyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2-methoxyethyl)-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-hydroxy-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
5-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}pyrimidin-2-amine
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
7-{7-methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[(3,4-dimethylphenyl)methyl]piperidin-3-ol
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2,3-dihydro-1-benzofuran-2-carboxamide
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-(1-ethyl-1H-pyrazole-3-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
ethyl 3-(2-phenylethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxylate
(1R,7S)-3-(2-ethylbutyl)-N-methyl-4-oxo-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{4-[(3-fluorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-(2,6-difluorophenoxymethyl)-N-[2-(2-methoxyphenyl)ethyl]-1,2-oxazole-3-carboxamide
N-(3-cyclopentylpropyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
1-methyl-4-{[3-(methylsulfanyl)phenyl]methyl}-2-phenylpiperazine
methyl 3-(5-methylthiophene-2-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)(methyl)[1-(pyridin-3-yl)ethyl]amine
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]propanoate
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
[1-(1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-methoxy-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
1-cyclopentanecarbonyl-N-[(1R)-2-hydroxy-1-phenylethyl]piperidine-4-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]propan-1-one
1-(2-methoxyphenyl)-3-{1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-1-(6-fluoro-2-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]ethane-1-sulfonamide
1-methyl-4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carbonyl]piperidine-4-carboxylate
N-(2-{7-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
methyl 2-{1-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]pyrrolidin-3-yl}acetate
(1R,3s,6r,8S)-4-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]-4-azatricyclo[4.3.1.13,8]undecane
2-(2,6-dimethoxypyridin-3-yl)-2-[ethyl(methyl)amino]acetic acid
1-[(2E)-2-methylbut-2-en-1-yl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-methyl-1,3-thiazole-4-carboxamide
2-{1-[(3-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3,5,6-trimethylpyrazine
5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
4-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}pyrimidine-5-carboxylic acid
1-{1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carbonyl]piperidin-3-yl}propan-1-one
1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
1-(5-{[benzyl(ethyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methylpiperidine-4-carbonyl)piperidine
4-oxo-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
3-(2-methyl-1H-imidazol-1-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
2-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-1-(morpholin-4-yl)ethan-1-one
2-methyl-6-({4-[4-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine