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N-(furan-2-ylmethyl)-4-{[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}pyridine-2-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-(cyclohexylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
{4-[5-(ethylsulfanyl)thiophene-2-carbonyl]-1,4-oxazepan-6-yl}methanol
(1R,5S,8R)-8-(dimethylamino)-N-[2-(3-methoxyphenyl)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(2-fluorophenyl)-3-phenylpropanamide
1-(2,2-dimethylpropyl)-3-{[ethyl(methyl)amino]methyl}-3-hydroxypiperidin-2-one
1-(2-oxo-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-4-(trifluoromethyl)pyrimidin-2-amine
8-cyclopropanecarbonyl-2-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2-chloro-4-fluorophenoxymethyl)-N-cyclohexyl-N-methyl-1,3-oxazole-4-carboxamide
7-(3-phenyl-1,2-oxazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-({4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}methyl)benzonitrile
3-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridin-1-ium-1-olate
3-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
N-[(3R,4S)-1-(cyclopropylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-4-acetamidobutanamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-(methylsulfanyl)-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,3-thiazole
3-[4-(4-chloro-2-hydroxybenzoyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
[(3-{2-[4-(furan-3-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
[3-({1-[4-(piperidin-1-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}naphthalene-2-carboxamide
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-methyl-2-[methyl(2-phenylethyl)amino]-N-(pyrazin-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-(2-fluorophenyl)-5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-amine
2-({5-[(4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2,3-dihydro-1H-isoindole
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[(3R)-pyrrolidin-3-yl]benzamide
N-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazine-1-carboxamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
N-[2-(2-methoxynaphthalen-1-yl)ethyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
2-methyl-7-[2-(4-methylphenoxy)ethanesulfonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-ethyl-4-(4-methyl-1H-imidazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2R,3S,6R)-5-cyclopentanecarbonyl-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(3aR,7aS)-2-[(4-fluoro-3-methoxyphenyl)methyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}thiomorpholine
3-oxo-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
N-(4-{4-[(2-hydroxybutyl)amino]piperidin-1-yl}phenyl)-5-phenylpentanamide
N-[3-(aminomethyl)-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl]pyridine-2-carboxamide
2-methyl-5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyrazine
1-benzyl-N3-cyclopropyl-N5-[(2-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(2-methoxyphenyl)methyl]-N-[(3-methyloxetan-3-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[4-(3-cyclopentylpropyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
1-(3-cyano-4-ethoxyphenyl)-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4-(4-methylphenoxy)piperidine
1-{4-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazin-1-yl}ethan-1-one
1-{[1-(2,5-dimethylphenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-(2,2-dimethylpropyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-{1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
1-(azocan-1-yl)-3-(5-{[(3-hydroxypropyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
8-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid