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N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-phenylcyclohexane-1-carboxamide
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N-butyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyrazine-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-(4-methylphenyl)-N-{3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}propanamide
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
(4aR,7aS)-4-(dimethyl-1,3-thiazole-5-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-({[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-N-methylbutanamide
5-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1H-indole
1-[2-(2-chlorophenyl)ethyl]-N-[(1-ethylpyrrolidin-2-yl)methyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[(2R)-oxolane-2-carbonyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-{[2-(2-benzamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-benzyl-1H-pyrazole-4-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
3-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)azetidin-3-yl]pyridine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyridin-3-yloxy)aniline
2-[5-(4-methanesulfonylphenyl)-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(2-methoxyethyl)-2,3-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]quinoxaline-6-carboxamide
1-(2-hydroxyethyl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
(3S,4S)-4-(morpholin-4-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-ol
5-{[(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}-N-(propan-2-yl)pyrimidin-2-amine
5-(2,4-difluorophenoxymethyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
ethyl 5-{[3-(2-ethyl-5-oxopyrrolidin-2-yl)propanamido]methyl}furan-2-carboxylate
1-cyclopentyl-N-(dicyclopropylmethyl)-N-methyl-6-oxopiperidine-3-carboxamide
N,N-dimethyl-6-{pyrazolo[1,5-a]pyridin-7-yl}pyridine-3-carboxamide
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-2-methoxyethan-1-one
3-(furan-2-yl)-1-{4-[(oxolan-3-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}propan-1-one
2-(4-fluorophenyl)-2-hydroxy-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(3-hydroxyphenyl)-N-methylacetamide
N,3,4,7-tetramethyl-N-[1-(pyridin-3-yl)propyl]-1H-indole-2-carboxamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
3-{5-[(2-chlorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
4-(4-chlorophenoxy)-1-[(3-methylphenyl)methyl]piperidine-4-carboxylic acid
ethyl 4-[(1-{4-[2-(3-chlorophenyl)acetamido]phenyl}piperidin-4-yl)amino]piperidine-1-carboxylate
2-(4-chloro-2-methylphenoxy)-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
4-[5-(1-cyclopropyl-1H-pyrrol-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]pyridine
methyl 3-[(3-hydroxy-4-methoxyphenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-{3-[(pyridin-3-yl)amino]propyl}acetamide
methyl 1-[4-(4-methylphenoxy)piperidine-4-carbonyl]pyrrolidine-2-carboxylate
ethyl 2-[1-(hydroxymethyl)-9-[(5-methylthiophen-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]acetate
2-[1-(4-chlorophenyl)-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
3-methyl-6-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyridazine
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-2,4-dimethoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
N-[1-(4-fluorophenyl)propyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-{4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carboxylic acid
methyl 1-[5-(2,4-difluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidine-4-carboxylate
2-cyclopropyl-5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-4-methylpyrimidine