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3-[(3R,4S)-1-[(3-methyl-1H-indol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-fluoro-3-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
2-ethyl-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
7-methyl-2-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(3-methoxyphenyl)-1-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]ethyl]-N,3-dimethylbutanamide
(2S,4S,5R)-4-{[2-(dimethylamino)ethyl]carbamoyl}-2-ethyl-5-(4-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
2-(3-chlorophenyl)-7-fluoro-3-[(4-methylpiperazin-1-yl)methyl]quinoline
methyl[(5-methyl-1H-indol-3-yl)methyl][(3-methylpyridin-2-yl)methyl]amine
7-cyclohexyl-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-{4-[6-amino-5-cyano-4-(1,5-dimethyl-1H-pyrazol-4-yl)pyridin-2-yl]phenoxy}acetic acid
N-(2-benzylphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
4-[2-(4-methylphenoxy)ethanesulfonyl]-2-(trifluoromethyl)morpholine
9-(3-cyclopentylpropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-hydroxy-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrrolidine-2-carboxamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-(2-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
1-(4-chlorophenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]cyclopropane-1-carboxamide
1-(adamantan-1-yl)-3-[2-(1-methylpiperidin-3-yl)ethyl]urea
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,1-dioxo-1λ6-thiane-4-carboxamide
(3R,4R)-3-cyclopropyl-1-(3,5-difluoropyridine-2-carbonyl)-4-methylpyrrolidin-3-ol
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]methylamine
2-methyl-2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)propane-1,3-diol
(1S,5R)-6-[(6-methoxy-2H-chromen-3-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-(3-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}propyl)morpholine
butyl N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
methyl 1-(2-methylpropyl)-5-[(3-phenylbutyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-oxo-8-[3-(thiophen-3-yl)propanoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-ethyl-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-[1-cyclopropyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
4-cyano-N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-1H-pyrrole-2-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
1-[(3S)-3-aminopyrrolidin-1-yl]-3-(azocan-1-yl)propan-1-one
5-acetyl-N,2,4-trimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrrole-3-carboxamide
N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(1S,5R)-6-(3-phenoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}morpholine-2-carboxamide
4-(4-fluorophenyl)-6-methylpyrimidin-2-amine
5-(1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1H-1,2,3-triazol-4-yl)pyrimidine
3-phenoxy-N-{1-[1-(prop-2-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propanamide
1-[4-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)phenyl]pyrrolidin-2-one
3-({1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
methyl 1-(2-methylpropyl)-5-[(2-methylpropyl)amino]-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-(2-phenylethyl)piperidin-3-yl}methanol
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)benzamide