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5-[(4-fluorophenyl)methyl]-5-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
(3R,9R)-11-(3,5-difluorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-methyl-N-(oxolan-3-ylmethyl)piperidin-4-amine
3-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]piperidine-1-carboxamide
N-[(2R,3R)-1'-[(2S)-2-hydroxy-2-phenylacetyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-methyl-N-(2-phenoxyethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
(3R,5S)-N-[2-(dimethylamino)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
3,5-dimethyl-4-{[2-(5-propylfuran-2-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
4-methoxy-N-methyl-3-(1H-pyrazol-3-yl)benzamide
2-[2-(2,5-dimethylphenyl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(4-methoxy-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-4-yl}acetamide
2-{3-[({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]piperidin-1-yl}ethan-1-ol
(1R,5R)-3-benzoyl-6-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(3R,4R)-4-(hydroxymethyl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-ol
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
N-({5-[(2-ethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2,6-dimethoxy-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-{1-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
5-acetyl-2,4-dimethyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-pyrrole-3-carboxamide
2-[3-(4-methoxyphenyl)-1-(3-methylbutyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2-[2-(pyridin-2-yl)ethyl]-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1-(2-phenylethyl)piperidin-2-one
4-[2-(methylsulfanyl)phenyl]-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{2-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
benzyl({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amine
5-cyclopropyl-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3-methyl-1H-pyrazole
4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{[cyclopropyl(6-methylpyridin-2-yl)methyl]carbamoyl}-1H-imidazole-4-carboxylic acid
(benzylsulfamoyl)[2-(pyrrolidine-1-sulfonyl)ethyl]amine
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
4-(cyclopropylmethyl)-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}quinoline
5-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
1-(2-fluorophenyl)-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
N-(1-benzylpiperidin-3-yl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
4-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N,N-dimethylpiperidin-3-amine
2-methyl-3-[(pyridin-3-ylmethyl)amino]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]benzamide
5-(2-chlorophenyl)-N-(oxan-3-ylmethyl)furan-2-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
8-methyl-N-[(4-methylphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(5-methoxy-2-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
5-tert-butyl-2-(oxolan-3-yl)-1H-1,3-benzodiazole
1-[(2-aminopyridin-3-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid