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5-[(4-benzylpiperidin-1-yl)methyl]-N-(2-hydroxyethyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[2-(3-chlorophenyl)ethyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
N-({5-[(4-chloro-3-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
2-[4-(2-aminophenyl)-1H-pyrazol-1-yl]-N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)acetamide
methyl 3-chloro-4-{[methyl(thian-4-yl)carbamoyl]amino}benzoate
N-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
3-(2-chlorophenyl)-3-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
({5-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-(2-ethoxypyridin-3-yl)-4-methoxybenzamide
1-{1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-2-methylpropan-1-ol
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-cyclohexylpropanamide
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-difluorobenzamide
N-[1-(4-{4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carbonyl}phenyl)-1H-pyrazol-4-yl]pyridine-3-carboxamide
methyl 3-acetamido-5-{[(4-ethylphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(2-chloro-4-fluorophenoxymethyl)-N-(3-ethoxy-2-hydroxypropyl)-1,2-oxazole-3-carboxamide
(1R,2S,9R)-11-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-(1-{4-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]phenyl}ethyl)acetamide
1-methyl-3-[1-(5-methylpyridine-3-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[1-(1-benzothiophene-5-carbonyl)piperidin-4-yl]ethyl}morpholine
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrrolidin-2-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(4-methylpyridin-3-yl)acetamide
5-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
2-(2-methylfuran-3-amido)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
(3aR,7aS)-2-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
7-(2,3-dihydro-1-benzofuran-2-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-N-[3-(morpholin-4-yl)propyl]-4-oxo-2-propyl-1,4-dihydropyridine-3-carboxamide
N-[(3S,4R)-1-(1,3-benzothiazole-6-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
N,N-dimethyl-3-[3-({[2-(pyridin-4-yl)ethyl]carbamoyl}amino)phenyl]propanamide
[2-({[2-(methoxymethyl)pyrimidin-5-yl]methyl}[(2-methylphenyl)methyl]amino)ethyl]dimethylamine
2-(butylsulfanyl)-6-{6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}pyrimidin-4-amine
2-({[2-(azepan-1-yl)ethyl](propan-2-yl)amino}methyl)benzoic acid
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2,5,6-trimethylpyrimidin-4-amine
1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine
3-(dimethyl-1,2-oxazol-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
1-(2-amino-4-{[(2-fluorophenyl)methyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-(methylamino)ethan-1-one
9-[2-(methylamino)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[(2S,4R,6S)-2-benzyl-6-(2-chloro-3-hydroxy-4-methoxyphenyl)oxan-4-yl]acetamide
2,6-dihydroxy-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]benzamide
N-[(1-benzylpiperidin-3-yl)methyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-benzyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-1,3-benzoxazole-5-carboxamide
N-[3-(3,4-dimethylphenoxy)propyl]-N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
2-[1-(5-methyl-4-phenylthiophene-3-carbonyl)pyrrolidin-2-yl]pyridine
1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
2-{2-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]phenoxy}ethan-1-ol
N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N-[2-(methylsulfanyl)ethyl]acetamide