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5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazole-3-carboxamide
(2S)-N-[2-(4-chlorobenzenesulfonamido)ethyl]-2-acetamido-4-methylpentanamide
ethyl[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl](1H-imidazol-2-ylmethyl)amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}acetamide
(3R)-1-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)pyrrolidin-3-ol
4-(2-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-2-yl}ethyl)phenol
1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
dimethyl(2-{2-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
1-(3-methoxyphenyl)-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
1-(1H-imidazol-2-ylmethyl)-4-(1-methylpiperidin-4-yl)piperazine
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[3-(1H-pyrazol-1-yl)propyl]amine
3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-2-phenylimidazo[1,2-a]pyridine
8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2,7-dimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]imidazo[1,2-a]pyridine-3-carboxamide
1-acetyl-N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]piperidine-4-carboxamide
1-(pyrimidin-2-yl)-N-[1-(thian-4-yl)piperidin-4-yl]piperidin-4-amine
3-methoxy-5-[({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)carbamoyl]benzoic acid
4-{3-[1-(3-methoxypropyl)-1H-pyrazol-3-yl]phenyl}-3-methylpyridine
2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]propane-1,3-diol
6-(2-chlorophenyl)-2-[3-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
5-ethyl-N-[(5-methylfuran-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-(4-fluorophenyl)-N-[1-(pyridin-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-(pyrrolidin-1-yl)propanamide
4-(3-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-4H-1,2,4-triazole
1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
6-(4-ethylphenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-({4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
(4aS,7aR)-1-(4-methyl-1H-pyrrole-2-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-oxo-1-(3-phenylpropyl)-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(2,3-difluorophenyl)methyl]piperidine-4-carboxamide
N-[4-(4-{[(3-fluorophenyl)methyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
4-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-{5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-1-yl}ethan-1-ol
5-acetyl-N-(1-{[(3,3-diphenylpropyl)carbamoyl]methyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
2-methoxy-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
3-{1-[1-(5-methylpyridin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenol
2-(4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-3-(1H-pyrazol-4-yl)propan-1-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(piperidin-1-yl)propan-1-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-5-ethylpyrimidin-2-amine
(benzylsulfamoyl)(methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
(1S,5R)-N-(2-methoxyphenyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole
2-[4-(2-chlorophenyl)phenoxy]-N-methylacetamide