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1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
5-(diethylamino)-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
[4-(2-phenylethyl)piperidin-4-yl]methanol
N-[(1-benzylpyrrolidin-3-yl)methyl]-5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-amine
(3S,4S)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-ol
4-{[3-(5,6-dimethylpyridin-2-yl)phenyl]methyl}morpholine
N3-[(4-methylphenyl)methyl]-4-oxo-N5-(oxolan-2-ylmethyl)-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopropyl-1-{2-[1-(quinolin-5-ylmethyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
(2E)-3-(4-methoxyphenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]prop-2-enamide
N-(2-{8-oxo-2-oxa-7-azaspiro[4.5]decan-7-yl}ethyl)pyridine-3-carboxamide
N-[2-(7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
2-ethyl-4-({2-[(3-methoxyphenyl)methoxy]phenyl}methyl)-1-methylpiperazine
(2R)-2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidine
6-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-(3-chlorophenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrazole
8-fluoro-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-[(3S,4R)-1-(2-ethoxyacetyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
(2R)-2-amino-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-phenylpropan-1-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
3-{4-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazin-1-yl}pyrazine-2-carbonitrile
N-benzyl-N-(cyclopropylmethyl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1,3-dimethyl-5-{2-oxo-2-[4-(9H-purin-6-yl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
2-{[2-(4-chlorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-({6-[4-(dimethylamino)phenyl]pyridin-3-yl}methyl)acetamide
5-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]-2,1,3-benzoxadiazol-1-ium-1-olate
N-[(2R,3R)-2-ethoxy-1'-(2,2,3,3-tetramethylcyclopropanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
methyl 3-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(2,4-dichlorophenyl)methyl]-3-(1H-imidazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(cycloheptylamino)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(3-methyloxetan-3-yl)methyl]-1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}urea
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N,5-dimethyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}acetamide
1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[3-(2-ethoxyethoxy)phenyl]-3-(2-hydroxypropan-2-yl)piperidine-1-carboxamide
N-[(2-methoxyphenyl)methyl]-4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
4-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[1-(2,6-dihydroxybenzoyl)piperidin-4-yl]pyrrolidin-2-one
2,3,5,6-tetramethyl-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]benzamide
(3-{4-[4-(propan-2-yl)piperazin-1-yl]phenyl}phenyl)methanol
2-(butylsulfanyl)-N4-{1-oxa-8-azaspiro[4.5]decan-3-yl}pyrimidine-4,6-diamine
[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
2,5-dimethyl-4-(4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrimidine
ethyl 8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
1-(2-methyl-5-oxo-1,4-diazepan-1-yl)-5-phenylpentane-1,5-dione
ethyl 1-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidine-4-carboxylate
5-[2-(furan-2-yl)azepane-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-{5-[(1R,3S)-3-aminocyclohexyl]-3-[(3,4-dimethoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid