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1-{2-[5-(thiophen-3-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
N'-cyclopentyl-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]butanediamide
2-{4-[(2,5-difluorophenyl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-methanesulfonylpropan-1-one
4-methyl-N-[(5-methylpyrazin-2-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-methyl-1-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}propan-1-one
3-(2-chlorophenyl)-3-{2-[4-(2,4-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)pyrrolidine-2,5-dione
3-(2-methoxyethyl)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylic acid
1-(4-chlorophenyl)-N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}cyclopropane-1-carboxamide
3-(methoxymethyl)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
8-[2-methyl-5-(1,2-oxazol-5-yl)benzenesulfonyl]-2,8-diazaspiro[4.5]decan-3-one
1-(3-methylpyridin-4-yl)-4-[4-(trifluoromethyl)benzoyl]-1,4-diazepane
N-({5-[(4-chloro-2-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
(3-{2-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-cyclopropyl-9-(6-methylpyrimidin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-{[methyl(oxolan-2-ylmethyl)amino]methyl}-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl][(2,3-difluoro-6-methoxyphenyl)methyl]methylamine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1H-pyrrole-3-carboxamide
6-(quinolin-3-yl)pyrazine-2-carboxylic acid
4-(4-chlorophenyl)-1-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]butan-1-one
2-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-[(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
benzyl(cyclobutylmethyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-[2-(4-methoxyphenyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(hydroxymethyl)-1-({2-[3-(morpholin-4-yl)propoxy]phenyl}methyl)pyrrolidin-3-ol
1-[(4-methylphenyl)methyl]-4-(2-phenylpyrimidine-5-carbonyl)piperazin-2-one
5-(1-benzoylpiperidin-4-yl)-3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrazine-2-carboxamide
1-(2-hydroxyethyl)-5-[(3-methoxyphenyl)methyl]-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
5-[(2-fluorophenyl)methyl]-5-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[3-methyl-1-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]acetamide
1-(2-{1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(1R,3S)-N-benzyl-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carboxamide
4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]sulfonyl}-1,3,5-trimethyl-1H-pyrazole
3-(1-benzyl-1H-imidazol-2-yl)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
8-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]-1,2,3,4-tetrahydroquinoline
4-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thiophene-2-sulfonamide
7-[(3S)-3-ethylmorpholine-4-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
4-ethyl-1-methyl-3-[1-(quinolin-4-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-N-phenylpyrimidin-2-amine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
4-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-N-cyclopentyl-4-oxobutanamide
1-[2-(4-chlorophenyl)morpholine-4-carbonyl]cyclopropane-1-carboxamide
1-(3-{[(1,3-benzoxazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)-3-[cyclohexyl(methyl)amino]propan-2-ol
N-[(1S,2R)-2-aminocyclobutyl]-6,7-diethoxy-3-methyl-1-benzofuran-2-carboxamide
5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
7-methyl-2-[6-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one