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ethyl 1-{5-[(cyclohexylmethyl)carbamoyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carbonyl}piperidine-3-carboxylate
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(3-oxopiperazin-1-yl)acetamide
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-1-[3-(methoxymethyl)pyrrolidin-1-yl]propan-1-one
N,N-dimethyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
4-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-(propan-2-yl)-1H-pyrazole
5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-N-{[5-(methoxymethyl)furan-2-yl]methyl}-4-methyl-1,3-thiazol-2-amine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(oxan-2-yl)ethyl]acetamide
methyl (2S,4R)-4-[3-(3-fluorophenyl)benzamido]-1-[(4-hydroxy-3-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-(4-{5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}thiophen-2-yl)ethan-1-one
methyl 3-{[(2,3-dimethyl-1H-indol-7-yl)formamido]methyl}-5-(furan-2-amido)benzoate
(1R,5S)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[2-(4-methylpiperazin-1-yl)propyl]-5,5-diphenylpiperidin-2-one
N-[(2-phenoxypyridin-3-yl)methyl]thian-4-amine
3-{[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)carbamoyl]amino}-2-methyl-N-(2-methylpropyl)benzamide
5-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamidoacetamide
[(4-{2-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
ethyl 2-[2-(3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)ethyl]-1,3-thiazole-4-carboxylate
N-benzyl-3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-N-methylpropanamide
(3aR,6aR)-2-(2-chloro-6-fluorobenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(2-hydroxy-4-methoxybenzoyl)-1-(4-methylphenyl)piperazin-2-one
2,4-dimethyl-6-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]pyrimidine
4-hydroxy-2-phenyl-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]pyrimidine-5-carboxamide
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-5-carboxamide
2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-5-methylpyrazine
ethyl 1-(2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)piperidine-4-carboxylate
3-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
(4aS,7aR)-1-(3-chloro-1,2-oxazole-5-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3,5-dioxomorpholin-4-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]acetamide
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-[(2,5-difluorophenyl)methyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
4-[(diethylamino)methyl]-5-ethyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]furan-2-carboxamide
1-(3-methoxypropyl)-3-{2-[3-(3-methylbutanoyl)piperidin-1-yl]-2-oxoethyl}-3-phenylpyrrolidine-2,5-dione
(1S,5R)-6-(2-ethoxyethyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzoic acid
1'-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(3S,4R)-3-(dimethylamino)-N-(3-fluorophenyl)-4-(4-methylphenyl)pyrrolidine-1-carboxamide
7-methyl-2-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
{3-[(3-chlorophenyl)methyl]-1-(1-methylcyclohexanecarbonyl)piperidin-3-yl}methanol
5-(azepane-1-carbonyl)-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{5-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]thiophen-2-yl}ethan-1-one
N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-9-methyl-9H-carbazole-3-carboxamide
4-(3-methylbutyl)-3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}piperazin-2-one
(2S,3R)-2-[({[(4-acetamidophenyl)methyl]carbamoyl}methyl)amino]-3-hydroxybutanamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(pyrazin-2-yl)pyrrolidin-3-yl]acetamide