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3-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
2-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-ethyl-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrimidin-2-amine
3-methyl-6-[5-(3-propyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]pyridazine
N-(2-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}propanamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
(1R,5S,8R)-8-methoxy-3-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-azabicyclo[3.2.1]octane
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylbenzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)piperidin-3-ol
2-({[(4-acetylphenyl)carbamoyl]amino}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-(propane-2-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[1-(hydroxymethyl)cyclopropanecarbonyl]-4-(pyridin-4-yl)-1,4-diazepan-6-ol
N,N-dimethyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
1-methyl-6-propyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
4-methyl-6-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyrimidin-2-amine
5-methoxy-N-[3-(4-methoxyphenoxy)propyl]-N-methylfuran-2-carboxamide
1-[4-(4-methyl-1,4-diazepane-1-carbonyl)phenyl]imidazolidine-2,4-dione
N-(1-phenylcyclopropyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(pyrrolidin-1-yl)ethan-1-one
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-methoxy-4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(5-ethylpyridin-2-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-methyl-N-[2-(morpholin-4-yl)ethyl]-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
6-(1-{[4-(1,2,3-thiadiazol-4-yl)phenyl]methyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
5-(4-benzylpiperidin-1-yl)-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole
2-{1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}propan-2-ol
4-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
N-[(2-fluorophenyl)methyl]-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,4-diazepan-5-one
[(1-cyclopentylpiperidin-4-yl)methyl][(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
1-[(5-ethylfuran-2-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
2-{3,9-diazaspiro[5.6]dodecan-9-yl}-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
4-methoxy-N-{1-[1-(4,4,4-trifluorobutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
4-[1-(adamantane-1-carbonyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
3-hydroxy-3-{[methyl(oxan-4-yl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-{2-[3-(cyclopropylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
6-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
N-cyclopropyl-4-acetamido-N-[(4-ethoxyphenyl)methyl]benzamide
N-cyclohexyl-3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-methylpropanamide
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methoxyphenol
1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}furan-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{methyl[2-(pyrrolidin-1-ylmethyl)propyl]amino}piperidin-1-yl)benzamide
(4aS,7aR)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-3-ethyl-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-methylpiperidin-4-ol
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[1-cyclohexyl-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol