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N-(butan-2-yl)-1-cyclopentyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[4-({[(5-chloro-2-methoxyphenyl)methyl](ethyl)amino}methyl)-3,5-dimethyl-1H-pyrazol-1-yl]ethan-1-ol
2-methyl-3-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}quinoxaline
7-[(4-methanesulfonylphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(4-methoxy-3-methylphenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
4-(5-ethyl-2-methylpyrimidin-4-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl (2R,4S)-4-hydroxy-1-[2-(prop-2-en-1-ylsulfanyl)acetyl]piperidine-2-carboxylate
6-methoxy-4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-({[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylacetamide
2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)acetamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(pyridazine-4-carbonyl)piperidin-3-yl]propanamide
7-(2-methoxyethyl)-2-(pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(2-ethyl-1H-imidazol-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}propanamide
1-(1-cycloheptylpiperidin-3-yl)-4-phenylpiperazine
1-cyclopropyl-N-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidine-3-carboxamide
methyl 2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetate
1-(2-methylpropyl)-4-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]pyrrolidin-2-one
1-[1'-(1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-{4-[4-(2-ethylpiperidine-1-carbonyl)phenoxy]piperidin-1-yl}-3-methoxypropan-1-one
N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-{[(1S,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenol
1-benzyl-5-(2-methylbutyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
4-chloro-1-methyl-3-(thiomorpholin-4-ylmethyl)-1H-indazole
[(3R,4R)-1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-(2-chloro-4-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}-6-methoxyphenoxy)acetic acid
6-(5-chloro-2-fluorobenzoyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
3-[4-(benzyloxy)piperidine-1-carbonyl]-1-(propan-2-yl)piperidine
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-pentanamidobenzamide
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]pyrazin-2-amine
2-(pyridin-2-yl)-7-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine-2-carboxylate
2-(2H-1,3-benzodioxol-5-yl)-8-methyl-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-ethyl-6-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-N-methylpyridine-3-carboxamide
N-{1-[4-(3-phenylpiperidine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}acetamide
1-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidine-3-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
ethyl 1-(2,4-difluorobenzoyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
1-[4-(thiomorpholin-4-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[1-(furan-3-ylmethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
2-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-4-(pyridin-3-yl)pyrimidine
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-4-chloro-1-methyl-1H-pyrazole
2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
4-(1H-imidazol-1-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
3-[(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
1-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-(1H-indol-3-yl)butan-2-yl]-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
6-oxo-N-(2-phenoxyethyl)-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
2-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-6-ethoxyphenol