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N-{2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-oxoethyl}methanesulfonamide
5-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-ylmethyl}-1,2,4-oxadiazole-3-carboxamide
4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(thiolan-3-yl)acetamide
1-({1-cyclohexyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-1,2-dihydropyridin-2-one
3-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenol
1-[4-(2,5-dimethoxybenzoyl)benzoyl]-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-[2-(1H-imidazol-4-yl)ethyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-(3-phenylpropyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(quinolin-2-ylmethyl)piperidin-4-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
N-[(3S,4R)-1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(2S,4R)-N-methyl-4-{[(4-phenylphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
(4S)-3,3,4-trimethyl-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-ol
4'-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(dimethylamino)-N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-methylpyrimidine-5-carboxamide
1-ethyl-N-[2-(4-fluorophenyl)ethyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-chloro-1-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
2-{[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]amino}ethan-1-ol
1-methyl-4-({1-[(4-phenylphenyl)methyl]piperidin-3-yl}methyl)piperazine
1-(1H-imidazole-4-carbonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-3-enamide
2,8-dimethyl-4-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]quinoline
(2S,4S)-4-cyclobutaneamido-N-ethyl-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]pyrrolidine-2-carboxamide
ethyl 1-{[1-(carbamoylmethyl)-1H-indol-3-yl]methyl}-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
4-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}piperazin-2-one
N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
2-(dimethyl-1,3-thiazol-4-yl)-N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)acetamide
methyl[(3-methylpyridin-2-yl)methyl]{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
(3S,4R)-3-benzyl-1-[(6-ethoxypyridin-3-yl)methyl]-4-methylpiperidin-4-ol
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
(2E)-1-[4-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)piperidin-1-yl]-3-phenylprop-2-en-1-one
1-[benzyl(methyl)amino]-3-[4-({[(3-chlorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
3-ethyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-1H-pyrazole-4-carboxamide
2-(1-cyclopentyl-4-{[4-(difluoromethoxy)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-(2-hydroxyethyl)-N-[(4-methylphenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
8-fluoro-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)quinoline-2-carboxamide
4-[3-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)butyl]-2-methoxyphenol
N-cyclopentyl-2-methyl-N-[(4-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)methyl]-1H-indole
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(4-methylpiperazin-1-yl)-N-[(1r,4r)-4-methoxycyclohexyl]benzamide
4-{[1-(3-methylthiophene-2-carbonyl)piperidin-2-yl]methyl}morpholine
6-(2-chlorophenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1,3-dimethyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-methoxyphenoxy)acetamide
(4aR,7aS)-1-(1H-imidazol-2-ylmethyl)-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione