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2-(furan-2-yl)-5-methyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1,3-oxazole
N-methyl-N-[2-(piperidin-1-yl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
5-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}phenyl)-2H-1,2,3,4-tetrazole
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-{[5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperidin-3-ol
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(dimethylamino)butan-1-one
4-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)thiomorpholine
4-[3-(diethylcarbamoyl)piperidin-1-yl]pyrimidine-5-carboxylic acid
N-{1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
7-(2-propyl-1H-imidazol-1-yl)-1,2-dihydroisoquinolin-1-one
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
N-(1-methoxybutan-2-yl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(1-methyl-1H-imidazol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
8-[(1-propyl-1H-imidazol-2-yl)methyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[(2-methylphenyl)methyl]-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-(propan-2-yl)-2-(4-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazin-1-yl)acetamide
8-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
5,6-dimethyl-2-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,3-benzodiazole
N-(furan-2-ylmethyl)-6-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-(2-hydroxy-2-phenylethyl)-N-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-4-oxo-1,4-dihydroquinoline-2-carboxamide
2-methoxy-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)quinoxaline
6-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
(1R,5R)-6-(cyclobutylmethyl)-3-(3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
6-methyl-3-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H-1,2,3-triazole
1-ethyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-(3-chlorophenyl)-N-methyl-3-phenylpropanamide
4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
(1S,9S)-11-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(3-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
N-(3-chloro-4-propanamidophenyl)-2,3-dihydro-1,4-benzodioxine-5-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
1-{[1-(3-fluorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-[1-(cyclohex-1-en-1-yl)ethyl]-3-(dimethyl-1,2-oxazol-4-yl)urea
1-(2-methoxyphenyl)-3-[1-(1-{spiro[2.5]octane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
4-(2-aminopyrimidin-4-yl)-7-(3,6-dimethylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-fluorophenyl)-2-{3-[3-(pyridin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(thiophen-2-ylmethyl)acetamide
N-methyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
(2S)-N-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-2-(morpholine-4-carbonyl)pyrrolidine-1-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(pyridin-2-yl)ethyl]benzamide
(2E)-1-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
3-[3-(methylsulfanyl)phenyl]pyrazolo[1,5-a]pyrimidine