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diethyl({3-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
3-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-{[4-(dimethylamino)oxan-4-yl]methyl}urea
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
3-hydroxy-3-[({imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)methyl]-1-(2-methoxyethyl)piperidin-2-one
5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-(dimethylamino)-N-(2-methyl-5-{[methyl(1-methylpiperidin-4-yl)carbamoyl]amino}phenyl)acetamide
3-(3-hydroxyphenyl)-1-[3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]propan-1-one
2-{2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
8-methyl-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
2-[1-({1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-amine
4-cyclopentyl-3-{2-oxo-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-8-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
4-benzyl-1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-ol
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylbenzamide
7-(cyclopropylmethyl)-2-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decane
5-(methoxymethyl)-N-(4-{5-methyl-4-[(naphthalen-2-ylformamido)methyl]-1,3-oxazol-2-yl}phenyl)furan-2-carboxamide
N-benzyl-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-[1-(2-methylphenyl)piperidin-4-yl]pyrrolidin-3-yl]methyl}piperidin-4-ol
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-ethylpyrrolidine-3-carboxamide
2-{3-[(diethylamino)methyl]-4-methoxyphenyl}-1H-1,3-benzodiazole-6-carboxylic acid
1-[1-(oxolane-3-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
N-methyl-6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazin-3-amine
N-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-methylcyclohexanamine
3-(diphenylmethyl)-N-[2-(furan-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[1-(3-chlorophenyl)-5-oxopyrrolidin-3-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(1S,5S)-N-[3-(trifluoromethyl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-{[ethyl(oxan-2-ylmethyl)amino]methyl}pyridin-2-amine
(2R,6S)-4-[6-(2-methoxyphenyl)pyridazin-3-yl]-2,6-dimethylmorpholine
N-methyl-N-[2-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]methanesulfonamide
methyl (2S,4R)-1-[2-(2,3-difluorophenyl)acetyl]-4-(dimethylamino)pyrrolidine-2-carboxylate
4-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl}benzoic acid
ethyl 2-(1-{1-[(2-methoxyphenyl)methyl]-5-[(3-methylbutyl)carbamoyl]-4-oxo-1,4-dihydropyridin-3-yl}-N-methylformamido)acetate
5-(4-methanesulfonylphenyl)-2-(1H-pyrrol-1-yl)pyridine
N-[2-(azepan-1-yl)ethyl]-2-(4-oxo-1,4-dihydroquinolin-1-yl)-N-(propan-2-yl)acetamide
N-benzyl-2-cyclopropyl-N-[(3-methylpyridin-2-yl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-methyl-6-(2-methylpropyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]pyrimidine-4-carboxamide
3-({4-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-methyl-2-(morpholin-4-yl)propyl]propanamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3,5-dimethylfuran-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(9H-purin-6-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-({[(2-benzyl-1,3-thiazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]furan-2-carboxamide
2-(2-methyl-1H-imidazol-4-yl)-N,N-bis(propan-2-yl)benzamide
N-{[3-methyl-7-(2-methyl-1,3-thiazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-(2-phenylethyl)pyrrolidin-2-one
3-{1-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)acetyl]piperidin-3-yl}benzoic acid
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl}){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
2-{1-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidin-3-yl}benzoic acid