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2-(5-{6-azaspiro[2.5]octan-1-yl}-1-cyclohexyl-1H-1,2,4-triazol-3-yl)acetamide
(2S)-1-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
4-(2-{[2-(2-methyl-1,3-thiazol-4-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzamide
2-(1H-pyrazol-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}butanamide
1-{2-hydroxy-3-[4-methoxy-2-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2,6-dimethylquinoline-3-carboxamide
2-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-1H-imidazole
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]pyrazine-2-carboxamide
4-(cyclopropylamino)-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
ethyl 3-benzyl-1-(pyridin-3-ylmethyl)piperidine-3-carboxylate
3-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-[3-(pyridin-3-yl)phenyl]urea
2-{1-[1-(propan-2-yl)piperidine-4-carbonyl]azetidin-3-yl}pyridine
[4-(5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenyl]methanol
(2S)-2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-3-phenylpropanamide
1-[1-cyclohexyl-3-(3,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
(4aS,7aR)-1-(3-chlorothiophene-2-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-4-amino-1-{[(1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]methanesulfonyl}-N-ethylpyrrolidine-2-carboxamide
1-(2-chlorophenyl)-4-{2-[4-(hydroxymethyl)phenyl]acetyl}piperazin-2-one
2-(2-ethyl-1H-imidazol-1-yl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-[2-ethyl-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carbonyl]piperidine-3-carboxylate
3-[({[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]pyrrolidin-3-ol
3-[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]propan-1-ol
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-1-methylpiperidine-2-carboxamide
ethyl 1-[5-(phenoxymethyl)-1H-pyrazole-3-amido]cyclobutane-1-carboxylate
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine-2-carboxamide
5-(cyclohexylamino)-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-(pyrrolidine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-(quinolin-7-yl)urea
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(5-ethylfuran-2-yl)methyl]pyrrolidin-3-yl]methanol
6-(hydroxymethyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-2-carboxamide
3-{[(2-chloropyridin-3-yl)methyl](methyl)amino}-1-(3-methylpiperidin-1-yl)propan-1-one
2-fluoro-N-{3-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-oxopropyl}benzamide
2-{1-[(3,4-difluorophenyl)methyl]-4-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
(1S,6R)-9-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-cyclobutyl-3-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]sulfamoyl}benzamide
methyl 2-{[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-4-(methylsulfanyl)butanoate
(5S,9aS,9bS)-5-[1-(3-methylphenyl)-1H-imidazol-2-yl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}acetic acid
2-(2-methoxyphenyl)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)acetamide
(2R,6S)-4-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylmorpholine
methyl 3-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(1-cycloheptylpiperidin-3-yl)cyclopent-1-ene-1-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
dimethyl(2-{1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)amine
2-{3-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
3-chloro-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
5-[1-(4-methylpentanoyl)piperidin-4-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
(3S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-fluoro-2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine