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1-(cyclopropylmethyl)-6-[(4-hydroxyphenyl)methyl]-3-[3-(1H-pyrazol-1-yl)phenyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{2-[1-(2-methoxyphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}acetamide
2-cyclopentyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
5-(propan-2-yl)-N-[2-(pyridin-2-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[4-({4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]piperazin-1-yl}methyl)-3-methyl-1H-pyrazol-1-yl]ethan-1-ol
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-methoxy-2-({[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}methyl)phenol
7-(1,2-oxazole-3-carbonyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(2-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-propoxyethan-1-one
2-(5-fluoro-2-methylphenyl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
1-[2-(dimethylamino)-4-{methyl[(3-methylpyridin-4-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-(2,2-dimethyloxan-4-yl)-N-ethyl-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(2-oxopiperidin-1-yl)propanoyl]piperidine-3-carboxylate
3-({[2-(2-chlorophenyl)ethyl]amino}methyl)pyrrolidin-3-ol
5-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]propanamide
2-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
1-[4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)thiophen-2-yl]ethan-1-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-3-(4H-1,2,4-triazol-4-yl)propan-1-one
2-ethyl-N-[3-(1H-indazol-1-yl)propyl]pyrimidine-5-carboxamide
4-benzyl-3-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}(benzyl)amino)propanamide
methyl N-{[(2S,4S)-4-fluoro-1-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]pyrrolidin-2-yl]methyl}carbamate
ethyl 3-{2-[4-(2-fluorobenzamido)-1H-pyrazol-1-yl]acetamido}-5-methylhexanoate
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
8-[(2,4-dimethoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(5-acetylthiophen-3-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-({4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
4-{[methyl(quinoxalin-2-ylmethyl)amino]methyl}-N-(1-methyl-1H-imidazol-2-yl)benzamide
5-{1-[2-(2,3-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
3-fluoro-4-(8-methoxy-2-methylquinolin-5-yl)benzene-1-sulfonamide
[(2-chloro-6-fluorophenyl)methyl](methyl)[2-(oxan-4-yl)ethyl]amine
(3S,4S)-1-(benzenesulfonyl)-4-[4-(2-fluorophenoxy)piperidin-1-yl]pyrrolidin-3-ol
N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-methylthiophene-2-carboxamide
methyl (2S,4R)-4-[5-(4-methoxyphenyl)furan-2-amido]-1-methylpyrrolidine-2-carboxylate
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-7-(methylsulfanyl)-3-{[(pyridin-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
4-ethyl-1-methyl-3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-(furan-2-yl)ethane-1,2-dione
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})amine
(1S,5R)-3-benzyl-6-(2-ethoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-1-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)urea
2-(ethylamino)-4-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1,3-thiazole-5-carboxamide
(1s,4s)-4-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]cyclohexan-1-ol
methyl 2-{[(2-fluorophenyl)methyl]sulfamoyl}-6-(4-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1S,5R)-6-(4-chloro-2-methylbenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-(1H-imidazol-4-yl)-N-(oxolan-2-ylmethyl)prop-2-enamide
methyl 2-(4-{[(oxan-3-ylmethyl)carbamoyl]amino}phenoxy)acetate