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(1S,5R)-3-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-2-[2-(5-phenylthiophen-2-yl)-1H-imidazol-1-yl]ethane-1-sulfonamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[4-(morpholin-4-yl)phenyl]methyl}acetamide
1-(2-methoxypyridine-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-[(3S,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-{[(2-hydroxy-3-methoxyphenyl)methyl]amino}ethyl)-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
9-[4-(1H-pyrazol-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-(diethylamino)-3-{4-[(4,4-dimethylpiperidin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
2-{[(1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
4-benzyl-3-ethyl-1-(1H-pyrazole-3-carbonyl)-1,4-diazepan-5-one
3-methoxy-1-[2-oxo-2-(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)ethyl]-1,2-dihydropyridin-2-one
(3S,4S)-4-cyclopropyl-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]pyrrolidine-3-carboxylic acid
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethan-1-one
{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,4-triazol-1-yl)propyl]amine
N-cyclopropyl-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
2-{[3-(3-chlorophenoxy)azetidin-1-yl]methyl}quinoline
2-(1H-1,3-benzodiazol-1-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
N-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
4-(3-fluorophenoxy)-1-(3-phenylpropyl)piperidine-4-carboxylic acid
4-({[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}methyl)-4-ethylhexanenitrile
ethyl 4-[1-(1H-indole-5-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
3-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]benzonitrile
2-amino-4-(5-hydroxy-2-methoxyphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
3-(3-propoxypiperidin-1-yl)-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazine
3-(1-methanesulfonylpiperidin-4-yl)-1-[3-(1,3-oxazol-5-yl)phenyl]urea
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(4,4,4-trifluorobutyl)amine
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-[3-(propan-2-yloxy)propyl]pyrrolidin-2-one
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-phenylazepane-1-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-chloro-N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-fluorobenzamide
2-cyclopropyl-5-[2-(3-methoxypropyl)piperidine-1-carbonyl]-4-methylpyrimidine
3-[(4-hydroxypiperidin-1-yl)methyl]-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
2-(2,4-dichlorophenoxy)-N-(oxan-3-ylmethyl)acetamide
(2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
3-fluoro-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyridine-4-carboxamide
(3S,9aR)-3-benzyl-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(1-benzofuran-2-yl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-1,2,4-triazin-3-amine
4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]phenol
N-[(4-methoxyphenyl)methyl]-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}-N-propylacetamide
5-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
N-(2-methoxyethyl)-5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-({6-[3-(piperazin-1-yl)phenyl]quinazolin-4-yl}amino)ethan-1-ol
N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylbutanamide
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(oxolan-2-ylmethyl)piperazine
1-benzyl-2-methyl-3-[2-(4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-4,5,6,7-tetrahydro-1H-indol-4-one