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N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-[2-(trifluoromethyl)phenyl]acetamide
5-fluoro-N,N-dimethyl-2-(1H-pyrazol-4-yl)pyrimidin-4-amine
1-(cyclopropylmethyl)-6-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
(2R)-2-amino-3-(ethylsulfanyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propanamide
{[5-(4-methoxyphenyl)furan-2-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]benzamide
2-(4-fluorophenyl)-2-hydroxy-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
2-(3-methylbutyl)-8-(pyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(1,2-oxazolidin-2-yl)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
5-{3-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
2-(1-methyl-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-phenoxypropan-1-one
N-[1-(thian-4-yl)piperidin-4-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
2-amino-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
methyl 5-[(adamantan-2-yl)amino]-3-acetamido-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-benzyl-N-(2-hydroxyethyl)-5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-4-carboxamide
methyl 3-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-(quinoline-8-sulfonamido)benzoate
8-chloro-2-({[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]amino}methyl)quinolin-4-ol
N-(3,5-difluorophenyl)-2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
1-{2-[(2-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-methylbutan-1-one
1-(2-aminopyrimidin-4-yl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylic acid
(1S,6R)-9-(4,6-dimethyl-2-oxo-2H-pyran-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
4-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
9-methoxy-7-(4-methoxyphenyl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{2-hydroxy-3-[4-methoxy-2-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
3-(1,3-dimethyl-1H-pyrazol-5-yl)-1-[3-(4-methylbenzenesulfonamido)propyl]urea
ethyl 3-[(2-methylphenyl)methyl]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
(3R)-1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3,4,4-trimethylpyrrolidin-3-ol
7-(2-methoxyethyl)-2-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-{[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
2,3-difluoro-5-(6-methyl-9H-purin-9-yl)phenol
3-{[4-(trifluoromethyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-ethyl-7-methoxy-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1H-indol-3-ylmethyl)(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
N-[1-(4-chlorophenyl)cyclobutyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-[1-(2-ethoxyethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-[(6-cyclopropylpyrimidin-4-yl)(methyl)amino]-1-phenylpropan-1-ol
8-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-1-oxa-8-azaspiro[4.5]decane
1-[2-(4-chlorophenyl)ethyl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
N-(3,5-dimethylphenyl)-N'-ethyl-N'-(pyridin-4-ylmethyl)propanediamide
3-cyclopentyl-1-({1-[(1-methylpiperidin-4-yl)methyl]piperidin-3-yl}methyl)urea
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-oxo-1,3-oxazolidine-4-carboxamide
2-(3-acetylphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(1-methyl-1H-indole-6-carbonyl)pyrrolidin-3-yl]methanol
2-(1-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}piperidin-4-yl)-N-methylacetamide