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N-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-propylpiperidin-3-amine
2-{[(5-methylpyrazin-2-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
2-(2-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}phenoxy)acetic acid
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1-azabicyclo[2.2.2]octan-3-amine
3-[4-(methylsulfanyl)benzoyl]-1-(1,2-oxazol-3-ylmethyl)piperidine
propyl 4-(4-benzyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxylate
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-hydroxy-3-methylbutan-1-one
1-(3,4-dimethoxyphenyl)-3-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]urea
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl][(2-methoxyphenyl)methyl]methylamine
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(2,5-dimethylthiophen-3-yl)-1H-pyrazol-1-yl]acetamide
4-(3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanoyl)-1,4-diazepane-1-carbaldehyde
2-chloro-5-acetamido-N-[(1-methylpiperidin-3-yl)methyl]benzamide
3-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-6-methyl-1,2-dihydroquinolin-2-one
(3S,4S)-4-cyclopropyl-1-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)pyrrolidine-3-carboxylic acid
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-(propan-2-yl)piperidine-3-carboxylic acid
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-methyl-N-(quinolin-2-ylmethyl)-1H-indazole-3-carboxamide
2-(1-ethylpiperidin-4-yl)-1-[1-(pyridin-3-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl]ethan-1-one
2-(3-{[4-(3-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}phenoxy)ethan-1-ol
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](thiophen-2-ylmethyl)amine
4-(4-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)-N-phenylpiperidine-1-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-[2-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3-methoxyphenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(4-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenoxy)pyrimidine
benzyl(ethyl){[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}amine
4-methyl-N-[3-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)propyl]benzene-1-sulfonamide
4-(1-cyclopentylpiperidine-4-carbonyl)-3-(1H-imidazol-4-ylmethyl)piperazin-2-one
7-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-3,4-dihydro-2H-1-benzopyran-4-one
ethyl 1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-3-carboxylate
1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)-4-(pyridin-3-ylmethyl)piperazine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-acetamidoacetamide
N,N-dimethyl-5-{[4-(4,6,7-trimethylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}-1,3-thiazol-2-amine
3-(4-methylphenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
1-(5-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-(oxolan-3-ylmethyl)acetamide
2-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1-benzofuran-5-carboxamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-(2-methoxyphenyl)propan-1-one
{5-methyl-7-[5-(1,2-oxazol-3-yl)thiophen-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3,7-dimethyl-11-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3,7,11-triazaspiro[5.6]dodecane
2-[4-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)morpholin-3-yl]-N-ethylacetamide
(3S,4R)-4-(2-methoxyphenyl)-1-[3-(pyridin-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-tert-butyl-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-[1-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-methyl-N-(2-phenylethyl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(benzenesulfonyl)-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine
6-({[1-(dimethylamino)cyclopentyl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-(2,6-dimethoxyphenyl)-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,3-triazole
3-chloro-N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)pyridine-4-carboxamide