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3-(furan-2-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
4-methyl-14-[2-(5-methylfuran-2-yl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-{1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-yl}piperidine
3-(1H-1,2,4-triazol-1-yl)-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
2-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
[5-({[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-(propan-2-yloxy)phenyl]methanol
N-[2-(dimethylamino)ethyl]-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[(5-methylthiophen-2-yl)methyl]benzamide
3-(2,6-dimethylhept-5-en-1-yl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(4aR,8aS)-6-[(4-methoxynaphthalen-1-yl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-propylpyrrolidin-3-yl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-butyl-1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]-2,5-dihydro-1H-pyrrole
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}acetamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
1-[3-(1,3-benzoxazol-2-yl)propyl]-3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)urea
6-[(furan-2-ylmethyl)amino]-N,N-dimethylpyridine-3-carboxamide
ethyl 5-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1H-1,3-benzodiazol-2-ylmethyl)({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
2-ethyl-5-({[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-1,3,4-oxadiazole
5-{4-[1-(furan-3-ylmethyl)pyrrolidin-3-yl]pyridin-2-yl}-8-methylquinoline
2-chloro-N-[2-(1,3-oxazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
4-{[(dimethylsulfamoyl)amino]methyl}-1-[(2-methyl-1,3-oxazol-4-yl)methyl]azepan-4-ol
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
2-methoxy-1-[1'-(trimethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-[2-(2-hydroxyphenyl)ethyl]-4-(2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-4-methyl-2-[(3-oxo-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl)amino]pentanamide
2-{[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-8-fluoro-3,4-dihydroquinazolin-4-one
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
N-({7-[2-(2,5-dimethoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(1H-imidazol-1-yl)acetamide
8-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
(1-benzofuran-2-ylmethyl)(1,4-dioxan-2-ylmethyl)methylamine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]piperazine
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-(pyridin-2-yl)piperazine
2-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-6-methyl-4H-pyran-4-one
6-{3-[methyl(phenyl)amino]propyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-ethyl-5-(3-fluoro-4-methoxyphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2,4-triazin-3-amine
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[3-(1H-imidazol-1-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-{1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-3-yl}benzoic acid
N,3,5,7-tetramethyl-N-[1-(pyridin-3-yl)propyl]-1H-indole-2-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-5-propyl-1,2-oxazole-3-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3-methylbenzoyl)pyrrolidin-3-yl]methanol
N-[2-methyl-4-(6-methyl-9H-purin-9-yl)phenyl]pyridine-3-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1-methyl-1H-pyrazole-5-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-5-(1-benzofuran-2-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[1-(adamantan-2-yl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
3-[2-(3-fluorophenyl)ethyl]-1-(oxane-4-carbonyl)piperidine