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N-(2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)acetamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[2-(pyrrolidin-1-yl)acetyl]-1,4-diazepan-5-one
dimethyl({2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]-1-(3-methylthiophen-2-yl)ethyl})amine
ethyl 1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
4-methyl-N-[2-(morpholin-4-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
5-acetyl-N-(1-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
methyl (2S)-1-{3-[2-(cyclohex-1-en-1-yl)acetyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}pyrrolidine-2-carboxylate
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenylpropanamide
3-{[(2,3-dihydro-1H-inden-4-yl)carbamoyl]methyl}-N-(propan-2-yl)morpholine-4-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-methyl-2-(propan-2-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
N-(4-chloro-2,6-dimethylphenyl)-2-(morpholin-4-ylmethyl)-1,4-oxazepane-4-carboxamide
2-amino-6-(3,5-difluorophenyl)-4-[2-(dimethylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
2-methoxy-4-[(1E)-3-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}prop-1-en-1-yl]phenol
N-methyl-6-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
4-(4-ethyl-6-{pyrazolo[1,5-a]pyridin-7-yl}pyrimidin-2-yl)morpholine
2-amino-4-{3-[(diethylamino)methyl]-4-methoxyphenyl}-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-methyl-N-(oxan-2-ylmethyl)-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
3-chloro-5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-ol
methyl({5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)(pyridin-3-ylmethyl)amine
N-{2-[(2-chlorophenyl)formamido]ethyl}-2-(morpholin-2-yl)acetamide
N-[(1-methylpiperidin-3-yl)methyl]-4-(2-oxopyrrolidin-1-yl)-N-(2-phenylethyl)butanamide
1-cyclopentyl-N-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
(1S,5R)-6-(propane-1-sulfonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-tert-butyl-N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
5-{[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}-2-methoxybenzoic acid
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
5-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenoxy}-1H-1,2,3,4-tetrazole
1-[3-(3-cyano-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)propyl]piperidine-4-carboxamide
3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
N-{4-[2-(dimethylamino)ethoxy]-1-(3-fluorophenyl)-1H-indazol-3-yl}-1H-1,2,4-triazole-5-carboxamide
4-{1-[2-(2-chlorophenyl)ethyl]-1H-imidazol-2-yl}benzamide
1-[(2-phenyl-1H-imidazol-4-yl)methyl]-4-(2-phenylethyl)piperazine
1-(3-{[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}propyl)pyrrolidin-2-one
N-(1-benzyl-5-oxopyrrolidin-3-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-hydroxy-5-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}benzoic acid
1-[(4,8-dimethoxynaphthalen-1-yl)methyl]-4-[2-(methylsulfanyl)ethyl]piperazine
N-{3H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{[(4aS,7aR)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
N-[(2,5-dimethylphenyl)methyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(3-methylbutyl)propanamide
4-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
2-{2-[4-(6-chloropyridin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4-methyl-6-(trifluoromethyl)pyrimidine
N-{[8-(2,6-dimethylhept-5-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-methoxyacetamide
8-{pyrazolo[1,5-a]pyrimidin-3-yl}-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-[(3-chlorophenyl)methyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-fluoro-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-methyl-1-benzofuran-2-carboxamide
[(3R,4R)-1-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
N-cyclooctyl-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-4-carboxamide