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1-(3-cyano-4-ethoxyphenyl)-3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]urea
6-{[(2S)-2-carbamoylpyrrolidin-1-yl]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(dimethylamino)-7-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
9-[2-(4-chlorophenyl)-2-hydroxyacetyl]-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
8-methoxy-2-(1H-pyrazol-4-yl)quinoline
N-[(2S,4R,6S)-2-benzyl-6-[(E)-2-phenylethenyl]oxan-4-yl]acetamide
2-[methyl(pyridin-4-ylmethyl)amino]-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
6-[(2,5-dimethylphenyl)methyl]-1-methyl-3-phenyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(3S,4R)-1-(cyclopentylmethyl)-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
1-(3-chlorophenyl)-5-methyl-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazin-2-one
6-fluoro-4-{4-[(pyrimidin-2-yl)amino]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
2-[2-(dimethylamino)ethyl]-9-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-cyclopentyl-6-oxopiperidine-3-carboxamide
1-[3-({1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}amino)piperidin-1-yl]ethan-1-one
4-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-(4-phenoxybenzoyl)piperidine
(1S,9aR)-1-({4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-octahydro-1H-quinolizine
3-butyl-4-(3-fluoropyridine-4-carbonyl)-1-methylpiperazin-2-one
N-methyl-3-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]pyridin-2-amine
5-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-2,4-dimethylpyrimidine
2-methoxy-N-(4-methyl-3-{[({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)carbamoyl]amino}phenyl)acetamide
1-cyclohexyl-4-[(2-hydroxy-6-methoxyphenyl)methyl]piperazin-2-one
1-[2-({[(2,4-difluorophenyl)methyl]amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
7-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-({5-[1-(cyclopentylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
[4-(5-methyl-1,3-diphenyl-1H-pyrazole-4-carbonyl)morpholin-2-yl]methanamine
8-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}quinoline-2-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
2-methyl-5-(3-methylphenyl)-4-[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]pyrimidine
methyl (2S)-1-{3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoyl}pyrrolidine-2-carboxylate
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(propylsulfanyl)acetamide
3-[({2-chloro-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}methyl)(methyl)amino]-N-methylbutanamide
N-butyl-3-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-methyl-N-[1-(pyridin-3-yl)pentyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl (2S)-2-({7-acetamido-1-[(4-fluorophenyl)methyl]-1H-1,3-benzodiazol-5-yl}formamido)-2-phenylacetate
3-(4-benzylpiperazine-1-carbonyl)-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
ethyl 2-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)acetate
N-(cyclopropylmethyl)-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-propylpropanamide
3-ethyl-4-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
3-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]-N-(2-fluoro-5-methylphenyl)propanamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(4-methyl-1H-imidazol-5-yl)-1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazole
N'-cyclopentyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]butanediamide
5-ethyl-3-{[5-(3-fluoro-5-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
4-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
ethyl 2-{1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-amido]cyclohexyl}acetate
N-methyl-2-(methylamino)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-4-carboxamide
2-methyl-4-(2-methylphenyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine