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4-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-5,6-dimethylpyrimidine
1-(carbamoylmethyl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}piperidine-4-carboxamide
3-{[benzyl(methyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
5-acetyl-3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
3-[1-(4-chloro-1H-indole-2-carbonyl)piperidin-3-yl]benzoic acid
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-difluorophenyl)acetamide
2-[1-({5-chloro-2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)azetidin-3-yl]pyridine
2-[4-(2-hydroxy-4-methoxybenzoyl)-2-oxopiperazin-1-yl]benzonitrile
N-[(3R,4S)-1-cyclopentanecarbonyl-4-(propan-2-yl)pyrrolidin-3-yl]-6-(methoxymethyl)pyrimidin-4-amine
N-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}-2,3-dimethoxy-N-(2-methoxyethyl)benzamide
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxamide
4-methoxy-N-{[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
ethyl 4-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
9-(isoquinolin-1-yl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
3-(2-methylpropyl)-6-(oxolan-3-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
5-[4-(4-methylphenyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}benzamide
2-{1-[(3-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
N-(2-hydroxyethyl)-2-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-dihydroquinoline-4-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
1-(pyridin-2-yl)-2-[(trimethylpyrimidin-4-yl)amino]ethan-1-ol
5-ethyl-5-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
1-(4-chloro-3-methylphenoxy)-3-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-2-ol
3-(4-fluorophenyl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-2,3-dimethoxy-N-(2-methoxyethyl)benzamide
2-methyl-8-{[2-methyl-5-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-cyclopentyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
2-{4-[(3-methoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-(4-methylphenyl)piperazine
N-(3-{4-[4-(2-ethoxyphenyl)piperazin-1-yl]piperidin-1-yl}phenyl)pyridine-3-carboxamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]acetamide
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-(3-hydroxypiperidin-1-yl)ethan-1-one
1-(2,6-dimethoxypyrimidine-4-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-methyl-5-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-[(2-fluorophenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{2-methyl-3-[({[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)methyl]-1H-indol-1-yl}acetamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N-methylpyrimidin-4-amine
2-[(2E)-hex-2-en-1-yl]-2,8-diazaspiro[4.5]decane
9-methoxy-7-(2-methoxyphenyl)-4-[(3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}-2,1,3-benzothiadiazole
2-[1-(2,2-dimethylpropyl)-4-[1-(2-methoxyphenyl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
(2S,4S)-4-amino-N-ethyl-1-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]pyrrolidine-2-carboxamide
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-methyl-3-(2-methylpropyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-{[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}quinolin-4-ol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,6-dimethyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-{[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
N-(3-hydroxypropyl)-3-(2-methyl-1H-imidazol-1-yl)-N-[(5-methylthiophen-2-yl)methyl]propanamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide