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3-(propan-2-yloxy)-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridazine
4-{[(2-methanesulfonamidoethyl)carbamoyl]amino}-N-(oxolan-2-ylmethyl)benzamide
6-[(3-ethoxy-2-hydroxyphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)ethan-1-one
6-[4-(4-fluorophenyl)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]propanamide
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-methyl-1-(3,4,5-trimethoxyphenyl)urea
2-[4-(2,1,3-benzoxadiazole-5-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
N-[1-(3-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methyl-1H-pyrazole-4-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(pyridin-4-yl)ethyl]piperidine-4-carboxamide
1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
N-({7-[(2E)-2-methylbut-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyrrolidine-1-sulfonyl)ethyl]amine
3-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-6-methoxyquinolin-2-ol
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(2-oxo-2-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)urea
1-(2,1,3-benzoxadiazol-4-ylmethyl)-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
N-[(1-propylpiperidin-3-yl)methyl]-2,3-dihydro-1H-inden-2-amine
2-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-4-methoxyphenol
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
5-{[methyl({3-[2-(4-{2-[3-(trifluoromethyl)phenyl]acetyl}piperazin-1-yl)ethoxy]phenyl}methyl)amino]methyl}pyrrolidin-2-one
ethyl 4-({[1-(1-methyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)benzoate
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(pyridazine-3-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
3,5,7-trimethyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-indole
3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
4-hydroxy-N-[(3-hydroxy-4-methoxyphenyl)methyl]-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
1-{1'-[(2,3-difluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]pyridine-4-carboxamide
N-(2-hydroxyethyl)-4-methyl-2-(pyridin-3-yl)-N-(thiophen-2-ylmethyl)pyrimidine-5-carboxamide
N2-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
4-methoxy-2-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[5-(propan-2-yl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-4-(4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}phenyl)butan-2-ol
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-tert-butyl-1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-[(3S)-1-benzylpyrrolidin-3-yl]propanamide
3-(2-methoxypyridin-3-yl)-1,5-dimethyl-1H-indazole
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(prop-2-en-1-yl)propanamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2-(piperidin-1-yl)-N-(pyridin-4-ylmethyl)acetamide
methyl (2S)-1-[1-(4-methylquinazolin-2-yl)piperidine-4-carbonyl]pyrrolidine-2-carboxylate
N-(furan-3-ylmethyl)-N-methyl-2,7-dioxo-1,3-diazepane-4-carboxamide
(2R,3S,6R)-3-(4-methylphenyl)-5-(1,3-thiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-3-(3-methoxyphenyl)propan-1-one
9-methoxy-7-(6-methoxypyridin-2-yl)-4-[2-(trifluoromethyl)benzenesulfonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
dimethyl({4-methyl-5-[1-(pyridine-3-sulfonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
5-methyl-5-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]morpholine