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N-methyl-N-[2-(oxan-4-yl)ethyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
(3aS,6aS)-2-cyclohexyl-5-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[(morpholine-4-carbonyl)amino]phenyl}-2-(thiomorpholin-4-yl)acetic acid
5-[2-(3-methoxyphenoxy)ethyl]pyridine-3-carboxamide
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-(3-phenylpropyl)-1,4-diazepane
(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
1-benzyl-4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-6-ol
(1S,5R)-3-benzyl-6-(4-chloro-2-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-{4-[(3,5-dichlorophenyl)methyl]morpholin-2-yl}ethyl)acetamide
4-methoxy-N-{[1-(3-methylbut-2-enoyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
methyl 3-(3-chlorobenzamido)-6-{[methyl(propan-2-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-methyl-5-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-3-carboxamide
3-[(3-methyl-1H-pyrazol-5-yl)formamido]-N-(naphthalen-1-yl)propanamide
2-[6-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-methylpyrimidin-4-yl]ethan-1-amine
(2S,4R)-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-methyl-1-(2-methylpropyl)pyrrolidine-2-carboxamide
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazine-1-carboxylate
1-[1-(2-aminoacetyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-6-(6-hydroxypyridine-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amine
1-ethyl-2-({2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1H-1,3-benzodiazole
(1R,2S,6R,7S)-4-(5-methoxy-1H-indazole-3-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
1,1,1-trifluoro-3-{3-[3-(pyridin-3-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
2-(oxan-2-ylmethyl)-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
1-{5-[(3,4-dichlorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}butan-2-ol
3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanoic acid
2-(7-fluoro-4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
4-{1-[2-(2-fluorophenyl)benzoyl]piperidin-3-yl}morpholine
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-[2-(pyridin-4-yl)ethyl]pyrrolidin-2-one
3-(1,2-oxazolidin-2-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
2-[2-(3-ethynylbenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
N-cyclohexyl-3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]propanamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-{3-[5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenyl}pyridine
ethyl 4-{6-[3-(5-methylfuran-2-yl)butyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-2,3-dihydro-1H-indene-1-carboxamide
3-(2,3-dimethylphenyl)-1-methyl-1-[2-(oxan-4-yl)ethyl]urea
3-{[(butan-2-yl)(3-phenylprop-2-yn-1-yl)amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
2-(3-methoxyphenyl)-1-{1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carbonyl}azetidine
1-(3-methylbutyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-acetylpiperazin-1-yl)-2-(5-fluoro-2-methylphenyl)acetic acid
2-[3-(2-methoxyphenoxy)azetidin-1-yl]-5-[(methylsulfanyl)methyl]pyridine
(2S,4R)-1-(2,6-difluoro-3-methylbenzoyl)-4-(dimethylamino)pyrrolidine-2-carboxylic acid
(1S,5R)-3-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{2-tert-butylimidazo[1,2-a]pyrimidin-3-yl}-3-methyl-1H-pyrazole
5-(azetidine-1-carbonyl)-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[(2R,3R)-1'-[(3-chloro-4-hydroxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-fluorobenzamide
{3-[(2,4-difluorophenyl)methyl]-1-(quinolin-4-yl)piperidin-3-yl}methanol
2-(2-methylphenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one