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3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
N-(1H-indol-4-ylmethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-{2-[(3-methyl-5-propyl-1-benzofuran-2-yl)formamido]ethyl}piperidine-3-carboxamide
(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-benzyl-3-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-phenylethane-1,2-dione
3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
2-chloro-4-({7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenol
2-{9-[(2R)-2,3-dihydroxypropyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-[({[7-methoxy-2-(thiomorpholin-4-yl)quinolin-3-yl]methyl}amino)methyl]cyclohexan-1-ol
2-tert-butyl-6-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)phenol
N-cyclopropyl-N-({4-[(2,5-dimethoxyphenyl)methoxy]phenyl}methyl)-3-methylthiophene-2-carboxamide
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[3-(cyclopentyloxy)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-{3-[1-(3-fluoropropyl)-1H-pyrazol-3-yl]phenyl}-4-methylpyridine
3-[(4-chlorophenyl)methyl]-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-[6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl]-3-(1H-pyrrol-1-yl)propan-1-one
3-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}benzoic acid
4-chloro-N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-(4-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)acetamide
1-cyclopentyl-4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazine
5-{[(5-methylpyrazin-2-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
[7-fluoro-5-(5-fluoro-2-methoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[1-(6-methoxynaphthalen-2-yl)ethyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
N-(2-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-cyclopentyl-N'-[(4-methylphenyl)(thiophen-2-yl)methyl]butanediamide
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
6-fluoro-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]-4-(pyrrolidine-1-carbonyl)quinoline
2-(2-methylphenyl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
N-(2-methyl-5-sulfamoylphenyl)thiomorpholine-4-carboxamide
1-(pyridin-2-yl)-N-(thian-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
3-[(ethylamino)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1-(4-{4-[(butan-2-yl)amino]piperidin-1-yl}phenyl)-5-methylpyrrolidin-2-one
(2S)-2-(dimethylamino)-N-[2-(4-methylphenyl)propan-2-yl]-3-phenylpropanamide
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-(quinolin-6-ylmethyl)propanamide
N-[(3-chlorophenyl)methyl]-2-[methyl(pyridin-3-ylmethyl)amino]-N-propylacetamide
N-(oxan-2-ylmethyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(methylsulfanyl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzamide
N-(2H-1,3-benzodioxol-5-yl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
2-amino-N-[2-(dimethylamino)ethyl]-N-methyl-1,3-benzothiazole-5-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
(1S,5R)-3-(5-acetyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-acetyl-1H-indol-1-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]butanamide
1-[3-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-[2-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
4-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-(oxolan-2-ylmethyl)-4-(4-{[4-(propan-2-yl)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione