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8-(1-benzofuran-2-sulfonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
3-methoxy-4-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
2-(3-methylphenyl)-5-{1-[1-(3-methylpyridin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
2-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1-(2-phenylphenyl)piperazin-2-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-methyl-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
2-cyclohexyl-6-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,3-benzoxazole
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]piperidin-4-amine
1-cycloheptyl-6-oxo-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
3-(azocan-1-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]propanamide
(1R,7S)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-oxo-3-[2-(piperidin-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-sulfamoyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
8-(2,4-difluoro-3-methoxybenzoyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-[5-(2-methyl-5-sulfamoylphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
4-{2,2-dimethyl-3-[4-(pyrazin-2-yl)piperazin-1-yl]propyl}morpholine
(3R,4R)-4-cyclopropyl-1-{[2-(difluoromethoxy)phenyl]methyl}-3-methylpiperidin-4-ol
5-(quinoline-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(thian-4-yl)piperazine
(3R,5R)-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
2-[ethyl(methyl)amino]-1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
5,5-dimethyl-3-{2-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-(3-methoxyphenyl)-N-(pyridin-3-ylmethyl)acetamide
(3-{3-[1-(2-methoxyethyl)-4-phenyl-1H-imidazol-5-yl]phenoxy}propyl)dimethylamine
N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-(2-methyl-4-{[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(prop-2-ene-1-sulfonyl)-decahydro-1,6-naphthyridin-2-one
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]pyrazine-2-carboxamide
1-(furan-2-ylmethyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
{3-[(3-chlorophenyl)methyl]-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}methanol
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}butan-1-one
N-methyl-2-(pyrrolidin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)benzamide
1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}pyrrolidin-3-amine
N2-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
2-{4-[(2-chloro-6-fluorophenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyrimidine
3-(4-benzylpiperidine-1-carbonyl)-2-ethyl-6-methyl-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridin-4-one
N-(2-{1-[(3-ethenylphenyl)methyl]piperidin-3-yl}ethyl)acetamide
N-(2-hydroxy-2-phenylethyl)-N-methyl-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
(4aS,8aR)-6-(1H-indole-6-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-3-ol
2-(4-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-({7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methoxybenzamide
3-({2-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{[3-methyl-7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide