提示: 按住Ctrl键可以同时选择多个官能团
1-{1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]piperidin-4-yl}pyrrolidin-2-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(propan-2-yl)piperidine-4-carboxamide
4-ethyl-3-[(1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
ethyl 2-[(5-{[4-(oxolane-2-carbonyl)piperazin-1-yl]methyl}pyrimidin-2-yl)amino]acetate
5-fluoro-N4,N4-dimethyl-N2-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-diamine
N-{1-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-methylpropyl}acetamide
1-(2-fluoro-4-methoxyphenyl)-2-(furan-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
4-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
5-acetyl-N-(1-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
1-[cyclohexyl(methyl)amino]-3-(2-{[(prop-2-en-1-yl)(prop-2-yn-1-yl)amino]methyl}phenoxy)propan-2-ol
1-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
7-methyl-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
5-[2-(6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(2-{[1-(carbamoylmethyl)piperidin-3-yl]formamido}ethyl)-4-fluorobenzamide
1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-2-(phenoxymethyl)-1H-1,3-benzodiazole
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
1-[3-(3-methylphenoxy)azetidin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
1-(4-phenylpiperazin-1-yl)-3-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]propan-1-one
(1S,5R)-3-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2E)-N-({7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(2-fluorophenyl)prop-2-enamide
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
4-(5-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-(3-fluorophenyl)-1-(7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-{[7-(furan-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-methoxybenzamide
3-[(3-ethyl-3-hydroxypiperidin-1-yl)methyl]-6-methyl-1,2-dihydroquinolin-2-one
1-(4-methyl-2-{[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]thiolan-3-amine
N-methyl-4-[(2-methylpyridin-3-yl)oxy]-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
2-[8-(2,2-dimethylpropyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
4,5-dimethyl-2-(2-methylpropanamido)-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]thiophene-3-carboxamide
(2S)-2-[(6-ethylpyrimidin-4-yl)amino]-3-phenylpropan-1-ol
2-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
2-[4-(furan-2-ylmethyl)piperazin-1-yl]-4-(pyridin-3-yl)pyrimidine
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(2-methylprop-2-en-1-yl)benzamide
(4-{[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
methyl 2-{8-[(3-methylthiophen-2-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
3-[({1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]piperidin-4-yl}amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
1-[6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl]-1,4-diazepan-5-one
2-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-N-tert-butylbenzene-1-sulfonamide
[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl][1-(2-fluorophenyl)propan-2-yl]amine
{2-[3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-2-oxo-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}urea
1-[2-(1H-imidazol-1-yl)ethyl]-4-(2-methoxynaphthalen-1-yl)-1H-1,2,3-triazole
2-[1-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperidin-4-yl]acetamide
N-({5-[(1-ethylpiperidin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide