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3-[(dimethylamino)methyl]-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-ol
{1-[7-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-2H-[1,3]dioxolo[4,5-g]quinolin-6-yl]piperidin-3-yl}methanol
N-cyclobutyl-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
3-(hydroxymethyl)-1-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}piperidin-3-ol
2-[(3,4-dimethoxyphenyl)methyl]-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
methyl({[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl})(quinolin-5-ylmethyl)amine
2-[1-(2,2-dimethylpropyl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-acetyl-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}thiophene-2-carboxamide
2,3-dimethoxy-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-3-yl)acetamide
4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1-methyl-2-phenylpiperazine
4-({[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
N-[(3-fluoro-4-methoxyphenyl)methyl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
(3aR,5S,6S,7aS)-2-(4-methoxy-3,5-dimethylbenzoyl)-octahydro-1H-isoindole-5,6-diol
methyl 6-[(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-3-carboxylate
1-[(4-chlorophenyl)methyl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-({4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
(2S)-1-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]pyrrolidine-2-carboxylic acid
N-[2-(morpholin-4-yl)ethyl]-4-{4-[(thiophen-3-ylmethyl)amino]piperidin-1-yl}benzamide
methyl 1-(3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-2-carboxylate
6-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
3-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
2-chloro-5-acetamido-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
[(4-methoxy-2,3-dimethylphenyl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
5-[(4-fluorophenyl)methyl]-3-(1-methylpiperidin-4-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2,6-dimethoxypyrimidine-4-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
(4aS,7aR)-1-(2-methyl-1,3-thiazole-5-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(2-phenylbenzoyl)piperidine
4,6-dimethoxy-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidine
9-[(2R,4S)-4-hydroxypyrrolidine-2-carbonyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl][4-(trifluoromethyl)phenyl]methanol
methyl 3-{[7-oxo-4-(2-phenylacetyl)-1,4-diazepan-1-yl]methyl}benzoate
1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
2-(2-hydroxyphenyl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonitrile
2-(1-benzyl-4-{[2-(furan-2-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
(3S,4R)-1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
6-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
benzyl 4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2-fluorophenyl)methyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(2R,6R)-4-[2-(2-oxoazepan-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}acetamide
methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]({5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amine
2-(2-fluoro-5-methoxyphenyl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
8-(5-chloropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]-1-(2-phenylethyl)pyrrolidin-2-one