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3-[(1-{2-[1-(propan-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propan-2-yl)oxy]pyridine
6-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-N,N-dimethylpyridine-3-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyridine-2-carboxamide
N-(1-{2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)acetamide
1-(2,5-dimethoxybenzoyl)-4-phenyl-1,4-diazepane
1-ethyl-3-methyl-N-[4-(5-methylfuran-2-amido)phenyl]-1H-pyrazole-4-carboxamide
[4-(1H-imidazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
7-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-methyl-N-[2-(morpholin-4-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-({7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methoxybenzamide
2-(1-benzyl-1H-pyrazol-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(2R,3R)-1'-(3-acetyl-1H-pyrazole-5-carbonyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(pyrrolidine-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-methanesulfonamido-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
N-[2-(dimethylsulfamoyl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(2,4-dichloro-6-methylphenyl)methyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-methoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-4-carboxamide
2-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]imidazo[1,2-a]pyrimidine-3-carboxamide
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
4-hydroxy-N-[3-(pyridin-4-yl)propyl]benzamide
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)acetamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(1H-pyrazol-1-yl)benzamide
N-{5-[3-(2-methoxyphenoxy)propyl]pyridin-2-yl}acetamide
N-(4-{4-[(cyclohexylformamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-5-(methoxymethyl)furan-2-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-ethyl-1H-pyrazole-3-carboxamide
(2R)-2-[(2-methyl-4-oxo-1,4-dihydroquinolin-8-yl)formamido]propanamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N2-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-N4-methylpyrimidine-2,4-diamine
(3S,4R)-1-(3-ethoxypropanoyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-2,3-dimethylquinoxaline-6-carboxamide
(2S,4S,5R)-1-methyl-2-(2-methylpropyl)-4-[(pyridin-2-ylmethyl)carbamoyl]-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
N-[2-(dimethylsulfamoyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(cyclohexylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(1,3-thiazol-2-ylmethyl)piperidin-4-ol
3-fluoro-N-{1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-butyl-5-(pyrrolidine-1-carbonyl)-1,3-benzoxazole
5-{[4-(2-methylpiperidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}isoquinoline
1-{6-hydroxy-4-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]-1,4-diazepan-1-yl}ethan-1-one
1-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N-(2-hydroxyethyl)-3-(2-hydroxyphenyl)-N-[(2-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
6-[9-(2-hydroxyethyl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyridine-2-carboxamide
6-{2-[(4-fluorophenyl)methyl]morpholine-4-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]furan-2-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide