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N-(2-methoxy-6-methylphenyl)-3-[(3-oxopiperazin-1-yl)methyl]benzamide
2-{6-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]pyrimidin-4-yl}ethan-1-amine
4-[(4-methoxyphenyl)methyl]-1-(4-phenylbutanoyl)-1,4-diazepan-5-one
5-[(2-fluorophenyl)methyl]-5-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
3-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}pyridin-2-amine
3-(4-hydroxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-3-(4-methoxyphenyl)-1H-pyrazole
(4aS,8aR)-6-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]pyridine
(2R,3R,6R)-5-(2-fluorobenzoyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-ethoxy-3-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-[(2-aminopyridin-3-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-(3-{2-[2-(propan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}propyl)-1H-1,3-benzodiazole
1-{4-[3-({[(6-methoxy-2H-chromen-3-yl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
ethyl 4-{1-[4-(thiophen-2-yl)butanoyl]piperidin-3-yl}piperazine-1-carboxylate
N-(2-phenoxyethyl)-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(1S,5R)-3-(2-ethylpyridine-4-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)cyclobutanecarboxamide
1-[(3,5-dimethylphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
3-[2-(2,6-difluorophenyl)ethyl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methylfuran-3-carboxamide
2-methanesulfonamido-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
(2S)-4-methyl-2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]pentanamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-methylazepane-2-carboxamide
4,5-dimethyl-6-[4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperazin-1-yl]pyrimidine
(2S,4R)-N-ethyl-4-(3-hydroxybenzamido)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
(1S,5R)-6-(4-fluoro-2-methylbenzoyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-4-propylpyrimidine-5-carboxamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one
1-(but-3-enoyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
methyl 7-oxo-9-(pyridin-4-ylmethoxy)-3-[4-(thiophen-2-yl)butanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[2-(thiophen-3-yl)acetyl]piperidin-3-yl]propanoic acid
4-(4-methyl-1H-pyrazol-1-yl)-1-(thiophen-2-ylmethyl)piperidine-4-carboxylic acid
N-[2-(4-methoxyphenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 1-{[4-(4-acetyl-1,4-diazepan-1-yl)quinazolin-2-yl]methyl}piperidine-2-carboxylate
6-(4-fluorophenyl)-7-methyl-8-oxo-N-{2-[(2R)-pyrrolidin-2-yl]ethyl}-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
7-cyclobutaneamido-N-[(3,5-difluorophenyl)methyl]-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
N-[(3S,4R)-1-[2-(4-ethoxyphenyl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-(3-phenyl-1H-pyrazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
2-{3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}pyridine
2-(4-fluoropiperidine-1-carbonyl)-5-methoxy-1,4-dihydropyridin-4-one
1-(carbamoylmethyl)-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]piperidine-3-carboxamide
1-(2-methyloxane-2-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
4-{5-[(2,4-dimethylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
N-(2-phenylethyl)-4-{[1-(thiophene-3-carbonyl)piperidin-4-yl]oxy}benzamide