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5-[1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
N-[(3-methylpyridin-2-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-dimethoxybenzamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1-phenylcyclopropane-1-carboxamide
N-(1-{4-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
7-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperidine
5-methoxy-1-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-indole-2-carboxamide
2-{1-[(6-methylpyridin-2-yl)methyl]-4-[(2,3,6-trifluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(1S,2R)-N1-(furan-2-ylmethyl)-N2-(prop-2-en-1-yl)-N1-(prop-2-yn-1-yl)cyclohexane-1,2-dicarboxamide
2-amino-1-{6-methyl-5-[5-(oxan-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}propan-1-one
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
[1-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
N-[4-(4-{[1-(pyridin-2-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
1-methyl-3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1-(thian-4-yl)urea
methyl 3-[(3S,4R)-1-[(4-fluorophenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
6-methyl-1-[(2-methylphenyl)methyl]-3-({[2-(pyridin-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-methyl-1,3,4-oxadiazol-2-amine
2-[4-(1-benzothiophen-3-yl)-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy]-1-[3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
2-[3-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)phenyl]ethan-1-amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-amine
5-fluoro-2-[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
5-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(naphthalen-1-yl)propan-2-yl]piperidin-4-amine
4-[6-oxo-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
1-(4-ethylpiperazin-1-yl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-methoxy-N-methyl-1H-indole-2-carboxamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
5-{[(3-chloro-2-fluorophenyl)methyl]carbamoyl}-1H-imidazole-4-carboxylic acid
3-{2-[3-(4-ethylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-(cyclopropylmethyl)-3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
7-methyl-2-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-acetyl-8-[2-(morpholin-4-yl)-2-oxoethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-benzyl-N-methyl-3-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)propanamide
N,N-dimethyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(2-methoxyphenyl)-2-methylpiperazine
3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
5-butyl-1'-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(1-methylpiperidin-2-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
2,7,8-trimethyl-4-[2-(1-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]quinoline
[(2,4-dimethoxy-3-methylphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
2-{[(1,3-benzoxazol-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrrole-3-carboxamide
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-N-(prop-2-en-1-yl)piperidine-1-carboxamide
5-(2-methoxyphenoxymethyl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
(3-{2-[1-(3-chlorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-hydroxy-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-1,2-oxazole-5-carboxamide