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[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)piperidin-3-yl]methanol
1-[(2,6-dichloro-3-hydroxyphenyl)methyl]-3-[(dimethylamino)methyl]piperidin-3-ol
1-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1H-pyrrol-1-yl)propan-1-one
N-(1,3-benzoxazol-2-ylmethyl)-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(2-methylbutanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-4-yl)piperidin-4-ol
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,4-dimethyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
2-{9-[(2-ethylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
(1R,3S,5S)-8-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
4-{1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidin-4-yl}pyridine
7-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-3-ol
(1-methyl-1H-imidazol-2-yl)(1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)methanol
3-(4-methoxypyridin-2-yl)-N,N-dimethylaniline
3-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-2-ol
1-cyclopentyl-N-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidine-3-carboxamide
(2S)-2-acetamido-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}propanamide
N-{4-[2-(methoxymethyl)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
1-{[4-(benzyloxy)phenyl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
(1S,4S)-2-(2,5-dimethoxyphenyl)-5-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-{2-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]propan-1-one
4-[2-(2-methoxyphenoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
1-{3-[2-(4-fluorophenyl)piperidine-1-carbonyl]phenyl}ethan-1-one
(4S)-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3,3,4-trimethylpiperidin-4-ol
6-[(3S,4R)-3-(propan-2-yl)-4-(2-propoxyacetamido)pyrrolidin-1-yl]pyridine-2-carboxylic acid
1-({4-[(2,3-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-N,N-diethylpiperidine-3-carboxamide
[(2-chloro-6-fluorophenyl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-(2-aminoethyl)-N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-6-(1H-1,2,3-benzotriazole-5-carbonyl)-1-butyl-decahydro-1,6-naphthyridin-2-one
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-phenylethane-1,2-dione
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]urea
(1R,5R)-6-(pyridin-2-ylmethyl)-N-(thiophen-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
7-methoxy-4-methyl-2-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}quinazoline
(3aS,6aS)-2-(2-chlorobenzoyl)-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}methanesulfonamide
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
4-{2-[(3-methoxyphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]propanamide
1-(4-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclobutanecarboxamide
N-(3-methoxypropyl)-N-{[2-(3-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carboxamide
8-(4-ethoxybenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2H-1,3-benzodioxol-5-yl)-2-[4-(1-methyl-1H-pyrazole-3-carbonyl)morpholin-3-yl]acetamide
1-methyl-4-({6-[2-(trifluoromethyl)phenyl]pyridin-3-yl}methyl)piperazine
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzene-1-sulfonamide
N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-1H-pyrrole-2-carboxamide