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N-[(2,6-difluoro-3-methylphenyl)methyl]-3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-ethyl-3-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-6-(cyclopropylmethyl)-3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-3-ol
4,4,4-trifluoro-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]butan-1-one
5-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
3-(2,4-dimethoxybenzoyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
4-{[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
2-tert-butyl-6-(3-methoxy-4-methylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-(4-methoxy-2-methylphenyl)-3-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}propanamide
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
methyl 4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}benzoate
3-(3-hydroxy-3-methylbutyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)benzamide
2-(4-{[4-(4-cyanophenyl)-3-oxopiperazin-1-yl]methyl}-2-methoxyphenoxy)acetamide
3-cyano-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)urea
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-ethoxypropan-1-one
(1S,5R)-N-benzyl-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
7-(3,5-dichloro-4-methylbenzoyl)-1-oxa-7-azaspiro[3.5]nonane
3-(3,4-dimethoxybenzoyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
6-fluoro-3-[2-(4-methylpiperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
2-amino-8-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
3-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)-3-phenylpyrrolidine-2,5-dione
3-methyl-N-[2-(pyridin-3-yloxy)propyl]furan-2-carboxamide
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-amine
3-(2-chlorophenyl)-N-methyl-N-[2-(pyridin-4-yl)ethyl]propanamide
N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(2-methanesulfonamidoethyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-benzyl-2-[1-cyclopentyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-(cyclopropylmethyl)acetamide
2-amino-6-(propan-2-yl)-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
2-(3-methoxyphenoxymethyl)-N-(1-phenylcyclopropyl)-1,3-oxazole-4-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-[4-(3-methoxyphenyl)phenyl]-1-(piperidin-4-yl)piperidine-3-carboxamide
1-(4-{[4-(benzyloxy)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-[(2R,3R)-2-(benzyloxy)-1'-(2,3-difluorobenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(3S)-1-[(1-{[1-(1,3-benzothiazol-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
4-(2-fluorophenoxy)-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
2-(dimethyl-1,2-oxazol-4-yl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)acetamide
N-[2-(dimethylamino)pentyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[6-methyl-3-({methyl[(3-methyloxetan-3-yl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
2-(2-methoxyphenoxy)-N-({1-[(3-methylphenyl)methyl]piperidin-3-yl}methyl)acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
ethyl 4-(3-phenylpropyl)-1-[3-(pyridin-3-yl)propanoyl]piperidine-4-carboxylate
3-[5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid