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2-methoxy-1-(4-{4-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
2-{[5-(dimethyl-1,3-oxazol-5-yl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{[4-(benzyloxy)phenyl]methyl}-1-(pyridin-2-ylmethyl)piperidin-3-amine
methyl 6-{[methyl(2-phenylethyl)amino]methyl}-3-(2-methylbutanamido)thieno[2,3-b]pyridine-2-carboxylate
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-methoxyphenyl)propanamide
N-(1-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
4-methoxy-N-[(2-methylphenyl)methyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
3-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
6-(cyclopropylmethoxy)-4-(furan-3-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
2-[methyl({5-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]ethan-1-ol
4-(4-fluorophenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-4-oxobutanamide
1-(2-methoxyethyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(1-methyl-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-yl)methanol
N-[1-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-methoxypropanamide
2-(1H-indol-5-yl)-N,6-dimethylpyrimidin-4-amine
3-methyl-3-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}urea
N-benzyl-1-ethyl-N-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-propyl-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]-2,5-dihydro-1H-pyrrole
4-fluoro-N-({1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl}methyl)benzamide
2-ethyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-({[(3R,4R)-1-[(3,5-dichloropyridin-4-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(2-methoxyphenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(thiophen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2,3-difluorophenyl)methyl]-4-[1-(1-methyl-1H-imidazole-5-carbonyl)pyrrolidin-3-yl]piperidine
N-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyridine-3-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-3-yl)propanamide
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
[1-({1-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-methyl-4-{4-[2-(pyridin-3-yl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
N-(5-hydroxypentyl)-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-4-carboxylate
(2R,6R)-4-[2-(2-oxopiperidin-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
8-fluoro-N-[1-(methylcarbamoyl)cyclohexyl]quinoline-2-carboxamide
3-[(cyclopentylamino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
4,6-dimethyl-2-{[1-(1-methylpiperidin-4-yl)piperidin-3-yl]amino}pyridine-3-carbonitrile
4-(1H-imidazol-1-yl)-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
4-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-1-cyclopropylpyrrolidin-2-one
3-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
6-[(4-methyl-1,4-diazepan-1-yl)methyl]-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
4-ethyl-3-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2,6-dimethyl-5-{2-[3-(3-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
(2S,4S)-4-amino-1-(3-cyclopentaneamido-4-methylbenzoyl)-N-ethylpyrrolidine-2-carboxamide
4-methyl-5-(2-phenylpyrrolidine-1-carbonyl)-1H-imidazole
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
3,5-dimethyl-7-(oxane-4-carbonyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
N,N-diethyl-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-4-carboxamide
2-(4-fluorophenoxy)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methylacetamide
N-(5-carbamoyl-2-fluorophenyl)-4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
4-({1-[3-(4-fluorophenyl)phenyl]piperidin-4-yl}amino)butan-1-ol